SCHEMBL3468423

SCHEMBL3468423

CC(COC(N)=O)c1ccc(Br)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.47
CYP1A2 P05177 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
CYP2D6 P10635 2/20 0.46
PKM P14618 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
EPHX1 P07099 2/20 0.41
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29213688 1.00 ALOX5 (0.47) ALOX5CYP1A2SMN1; SMN2CYP2D6PKM
SCHEMBL4590669 0.82 CYP1A2 (0.68) ALOX5CYP1A2SMN1; SMN2CYP2D6PKM
SCHEMBL28958757 0.82 CYP1A2 (0.68) ALOX5CYP1A2SMN1; SMN2CYP2D6PKM
SCHEMBL4589554 0.82 CYP1A2 (0.68) ALOX5CYP1A2SMN1; SMN2CYP2D6PKM
SCHEMBL27860265 0.81 CYP1A2 (0.43) ALOX5CYP1A2SMN1; SMN2CYP2D6NPSR1
SCHEMBL25254767 0.81 PKM (0.49) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL28989195 0.81 CYP1A2 (0.47) ALOX5CYP1A2SMN1; SMN2CYP2D6PKM
SCHEMBL14966967 0.80 ALOX5 (0.51) ALOX5CYP1A2SMN1; SMN2EPHX1MEN1
SCHEMBL6223098 0.80 ALOX5 (0.51) ALOX5CYP1A2SMN1; SMN2EPHX1MEN1
SCHEMBL20563823 0.80 CYP1A2 (0.56) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117820236-A Histone acetyltransferase small molecule inhibitor and preparation method and application thereof 复旦大学 2024-04-05 CN disclosed
WO-2010075270-A1 4, 6-DISUBSTITUTED 2-AMINO-PYRIMIDINES AS HISTAMINE H4 RECEPTOR MODULATORS INCYTE CORPORATION (US) 2010-07-01 WO disclosed