SCHEMBL3468432

SCHEMBL3468432

Cc1ccc(-c2ccc(C#N)cc2)cc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.46
MMP3 P08254 1/20 0.45
MAP4K4 O95819 1/20 0.45
ALDH1A1 P00352 4/20 0.45
CYP2A6 P11509 1/20 0.45
TDP1 Q9NUW8 2/20 0.43
CYP3A4 P08684 2/20 0.43
CASP1 P29466 1/20 0.43
TSHR P16473 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
KDM4E B2RXH2 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD11B1 P28845 2/20 0.40
EGLN2 Q96KS0 2/20 0.40
HRH3 Q9Y5N1 1/20 0.40
HRH4 Q9H3N8 1/20 0.39
GABRA1 P14867 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31757929 1.00 KIF11 (0.46) KIF11MMP3MAP4K4ALDH1A1CYP2A6
SCHEMBL21388680 0.85 ALDH1A1 (0.65) KIF11MMP3MAP4K4ALDH1A1CYP2A6
SCHEMBL29502034 0.84 ALDH1A1 (0.50) ALDH1A1CYP2A6TDP1CYP3A4CASP1
SCHEMBL178452 0.84 ALDH1A1 (0.50) ALDH1A1CYP2A6TDP1CYP3A4CASP1
Hydrochloric Acid SCHEMBL6476027 0.82 ALDH1A1 (0.48) ALDH1A1CYP2A6TDP1CYP3A4CASP1
SCHEMBL10304732 0.82 KIF11 (0.50) KIF11MMP3MAP4K4ALDH1A1CYP2A6
SCHEMBL15156687 0.82 TDP1 (0.61) KIF11MMP3MAP4K4ALDH1A1CYP2A6
SCHEMBL29655663 0.82 TDP1 (0.61) KIF11MMP3MAP4K4ALDH1A1CYP2A6
SCHEMBL6866139 0.81 CYP3A4 (0.62) ALDH1A1TDP1CYP3A4CASP1TSHR
SCHEMBL31661348 0.81 CYP3A4 (0.62) ALDH1A1TDP1CYP3A4CASP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010085968-A1 TOLUIDINE SULFONAMIDES AND THEIR USE AS HIF-INHIBITORS EUROPEAN MOLECULAR BIOLOGY LABORATORY (EMBL) (DE) 2010-08-05 WO disclosed
WO-2010076034-A1 TOLUIDINE SULFONAMIDES AND THEIR USE AS-INHIBITORS EUROPEAN MOLECULAR BIOLOGY LABORATORY (EMBL) (DE) 2010-07-08 WO disclosed