SCHEMBL3470000

SCHEMBL3470000

C/C=N/N(C)c1cc(=O)n(Cc2ccccc2)c(=O)[nH]1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.49
ALDH1A1 P00352 5/20 0.49
KDM4E B2RXH2 3/20 0.49
THRB P10828 2/20 0.49
SMN1; SMN2 Q16637 3/20 0.44
LMNA P02545 2/20 0.43
CYP3A4 P08684 1/20 0.43
PKM P14618 1/20 0.42
GAA P10253 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3473567 0.79 HPGD (0.51) HPGDALDH1A1KDM4ESMN1; SMN2CYP3A4
SCHEMBL3475882 0.79 TSHR (0.44) HPGDALDH1A1KDM4ETHRBSMN1; SMN2
SCHEMBL2182131 0.76 SMN1; SMN2 (0.61) HPGDALDH1A1KDM4ETHRBSMN1; SMN2
SCHEMBL2182128 0.76 SMN1; SMN2 (0.61) HPGDALDH1A1KDM4ETHRBSMN1; SMN2
SCHEMBL6518554 0.76 HPGD (0.51) HPGDALDH1A1KDM4ESMN1; SMN2LMNA
SCHEMBL6518558 0.76 HPGD (0.51) HPGDALDH1A1KDM4ESMN1; SMN2LMNA
SCHEMBL3471954 0.74 ALDH1A1 (0.62) HPGDALDH1A1KDM4ETHRBSMN1; SMN2
SCHEMBL3470482 0.73 ALDH1A1 (0.63) HPGDALDH1A1KDM4ETHRBSMN1; SMN2
SCHEMBL6243233 0.70 KMT2A (0.55) HPGDALDH1A1KDM4ESMN1; SMN2CYP3A4
SCHEMBL6247418 0.69 ALDH1A1 (0.53) HPGDALDH1A1KDM4ESMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010072807-A2 INHIBITORS OF CYSTATHIONINE BETA SYNTHASE TO REDUCE THE NEUROTOXIC OVERPRODUCTION OF ENDOGENOUS HYDROGEN SULFIDE FONDATION JEROME LEJEUNE (FR) 2010-07-01 WO disclosed
WO-2010072807-A2 INHIBITORS OF CYSTATHIONINE BETA SYNTHASE TO REDUCE THE NEUROTOXIC OVERPRODUCTION OF ENDOGENOUS HYDROGEN SULFIDE FONDATION JEROME LEJEUNE (FR) 2010-07-01 WO disclosed