SCHEMBL3471909

SCHEMBL3471909

COc1cc(N)c(C(C)C)cc1OC.COc1cc(N=C=O)c(C(C)C)cc1OC

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
CYP3A4 P08684 1/20 0.43
HPGD P15428 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
GAA P10253 2/20 0.40
POLB P06746 1/20 0.40
GFER P55789 1/20 0.40
P2RX3 P56373 10/20 0.35
P2RX2 Q9UBL9 10/20 0.35
KDM4E B2RXH2 1/20 0.34
PKM P14618 1/20 0.34
MGAM O43451 1/20 0.31
SI P14410 1/20 0.31
MGAM2 Q2M2H8 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1099288 0.91 CYP3A4 (0.50) ALDH1A1CYP3A4HPGDTDP1GAA
SCHEMBL3471609 0.91 CYP3A4 (0.50) ALDH1A1CYP3A4HPGDTDP1GAA
SCHEMBL1099448 0.80 GAA (0.55) ALDH1A1CYP3A4TDP1GAAPOLB
SCHEMBL28014621 0.76 ALDH1A1 (0.56) ALDH1A1CYP3A4HPGDTDP1GAA
SCHEMBL28573888 0.75 CYP3A4 (0.41) ALDH1A1CYP3A4HPGDTDP1GAA
SCHEMBL3478142 0.73 ALDH1A1 (0.45) ALDH1A1CYP3A4HPGDTDP1POLB
SCHEMBL29631745 0.71 GAA (0.58) ALDH1A1CYP3A4HPGDTDP1GAA
SCHEMBL6372278 0.71 CYP3A4 (0.63) ALDH1A1CYP3A4HPGDTDP1POLB
SCHEMBL542663 0.71 CYP3A4 (0.68) ALDH1A1CYP3A4HPGDTDP1POLB
SCHEMBL20755697 0.69 P2RX3 (0.55) ALDH1A1GAAPOLBGFERP2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393781-A1 DIHYDROPYRIDONE UREAS AS P2X7 MODULATORS F. Hoffmann-La Roche AG (CH) 2011-12-14 EP disclosed
WO-2010072599-A1 DIHYDROPYRIDONE UREAS AS P2X7 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2010-07-01 WO disclosed