SCHEMBL3476013

SCHEMBL3476013

COc1c(N)cc(F)cc1CCCC=O

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.33
CYP1A2 P05177 1/20 0.33
CYP19A1 P11511 1/20 0.33
IMPDH2 P12268 1/20 0.31
ABCB1 P08183 1/20 0.30
ABCC1 P33527 1/20 0.30
ALOX5 P09917 1/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30
CA14 Q9ULX7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10751588 0.85 CYP1A2 (0.41) HTR2ACYP1A2ALOX5CA12CA1
SCHEMBL2412839 0.78 POLB (0.41) IMPDH2
SCHEMBL18304159 0.77 PTGS2 (0.39) HTR2ACYP19A1ABCB1ABCC1
SCHEMBL2138518 0.74 TNF (0.43) CYP1A2
SCHEMBL3477926 0.74 CXCR2 (0.31)
SCHEMBL2689430 0.74 SLC6A2 (0.48)
SCHEMBL30504065 0.73 CYP19A1 (0.59) HTR2ACYP19A1ABCB1CA12CA1
SCHEMBL10750374 0.71 MEP1B (0.39) CA12CA1CA2CA14
SCHEMBL9963467 0.71 CYP19A1 (0.35) CYP19A1ABCB1ABCC1
SCHEMBL2689802 0.70 SLC6A2 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120101134-A1 5-MEMBERED HETEROARYL DERIVATIVES USED AS SPHINGOSINE 1-PHOSPHATE RECEPTOR AGONISTS GLAXO GROUP LIMITED (GB) 2012-04-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120101134-A1 5-MEMBERED HETEROARYL DERIVATIVES USED AS SPHINGOSINE 1-PHOSPHATE RECEPTOR AGONISTS S1PR1, S1PR5, S1PR3 HTR2A 404/4885CYP1A2 2262/4885CYP19A1 2930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.