SCHEMBL3476293

SCHEMBL3476293

NC(=O)c1cccnc1-c1cc(C(F)(F)F)ccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.44
RPS6KB1 P23443 2/20 0.44
AURKB Q96GD4 1/20 0.44
PARP1 P09874 4/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.42
LMNA P02545 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
MEN1 O00255 1/20 0.42
GMNN O75496 1/20 0.42
TTR P02766 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
PKM P14618 1/20 0.42
NFKB1 P19838 1/20 0.42
UGT1A1 P22309 1/20 0.42
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
PMP22 Q01453 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15903182 0.83 AURKA (0.51) AURKARPS6KB1AURKBPARP1KDM4E
SCHEMBL1968501 0.82 BCAT2 (0.46) AURKARPS6KB1AURKBPARP1KDM4E
SCHEMBL5178386 0.81 PARP1 (0.58) AURKARPS6KB1AURKBPARP1KDM4E
SCHEMBL5665026 0.78 TRPV1 (0.52) PARP1TRPV1CASP1
SCHEMBL17895180 0.78 TLR7 (0.46) AURKAKDM4EKMT2ANOS3NOS2
SCHEMBL3620548 0.76 GRM5 (0.51) PARP1KDM4EALDH1A1LMNATDP1
SCHEMBL4186883 0.75 KDM4E (0.65) PARP1KDM4EALDH1A1LMNATDP1
SCHEMBL27910329 0.74 SYK (0.53) AURKAKDM4EDHODHSYK
SCHEMBL29455925 0.74 GRM5 (0.50) PARP1KDM4EALDH1A1LMNATDP1
SCHEMBL28994207 0.74 AURKA (0.44) AURKARPS6KB1AURKBPARP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010034838-A2 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO claimed