SCHEMBL3476309

SCHEMBL3476309

Cc1ccc(-c2c(CC(=O)O)c(C)nc3sc4ccccc4c23)cc1

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.61
SMN1; SMN2 Q16637 1/20 0.54
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47
KDM4E B2RXH2 2/20 0.46
DPP4 P27487 2/20 0.45
EGLN1 Q9GZT9 1/20 0.42
MEN1 O00255 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
GFER P55789 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99124 0.88 KMT2A (0.48) KMT2ASMN1; SMN2KDM4EDPP4EGLN1
SCHEMBL15875874 0.87 KMT2A (0.47) KMT2ASMN1; SMN2LMNAPOLBDPP4
SCHEMBL99422 0.83 KMT2A (0.65) KMT2ASMN1; SMN2LMNAPOLBKDM4E
SCHEMBL134762 0.82 KMT2A (0.43) KMT2A
SCHEMBL99267 0.81 KMT2A (0.65) KMT2ASMN1; SMN2LMNAPOLBDPP4
SCHEMBL27709824 0.81 SMN1; SMN2 (0.43) KMT2ASMN1; SMN2LMNAKDM4EEGLN1
SCHEMBL99980 0.79 KMT2A (0.63) KMT2ASMN1; SMN2DPP4
SCHEMBL134802 0.79
SCHEMBL4056576 0.78 SMN1; SMN2 (0.40) KMT2ASMN1; SMN2KDM4EEGLN1GAA
SCHEMBL16109055 0.77 KMT2A (0.55) KMT2ASMN1; SMN2LMNAPOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9499563-B2 Thieno [2, 3-B] pyridine derivatives as viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2016-11-22 US claimed
US-20140296272-A1 THIENO [2, 3-B] PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS CISTIM LEUVEN VZW (BE) 2014-10-02 US claimed
EP-2430029-B1 THIENO[2,3-B]PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS UNIV LEUVEN KATH (BE) 2018-01-10 EP disclosed
US-9499563-B2 Thieno [2, 3-B] pyridine derivatives as viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2016-11-22 US disclosed
US-20140296272-A1 THIENO [2, 3-B] PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS CISTIM LEUVEN VZW (BE) 2014-10-02 US disclosed
US-8785638-B2 Thieno [2, 3-B] pyridine derivatives as viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2014-07-22 US disclosed
WO-2010130842-A1 THIENO [2, 3-B] PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2010-11-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140296272-A1 THIENO [2, 3-B] PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS TYMP, DUT, MAVS KMT2A 2903/4885SMN1; SMN2 3831/4885LMNA 3907/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.