SCHEMBL3477071

SCHEMBL3477071

COc1ccc(Cn2cc(B(O)OC(C)(C)C(C)(C)O)cn2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.43
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
PDE1A P54750 1/20 0.37
PDE1B Q01064 1/20 0.37
PDE1C Q14123 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
KLKB1 P03952 1/20 0.37
RET P07949 1/20 0.36
ERCC5 P28715 1/20 0.36
AADAT Q8N5Z0 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
NPBWR1 P48145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL594119 0.87 L3MBTL1 (0.43) L3MBTL1KLKB1ADORA2AADORA1MAPT
SCHEMBL455008 0.79 KMT2A (0.30) KMT2A
SCHEMBL15663094 0.77 IKBKE (0.32) RET
SCHEMBL4208996 0.76 L3MBTL1 (0.40) L3MBTL1
SCHEMBL2377232 0.75 FFAR1 (0.32)
SCHEMBL15663128 0.75
SCHEMBL2631271 0.75 ACHE (0.41)
SCHEMBL366006 0.75 CA1 (0.52)
SCHEMBL27901467 0.75 L3MBTL1 (0.53) L3MBTL1HSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL26622753 0.75 L3MBTL1 (0.49) L3MBTL1HSP90AA1HSP90AB1PDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010070076-A1 ALKANOIC ACID DERIVATIVES AND THEIR THERAPEUTIC USE AS HDAC INHIBITORS CRYSTAX PHARMACEUTICALS, S.L. (ES) 2010-06-24 WO disclosed