SCHEMBL3484150

SCHEMBL3484150

Nc1ccc(Oc2ccn3nccc3c2)c(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.38
DRD4 P21917 2/20 0.38
DRD3 P35462 2/20 0.38
PDE7A Q13946 1/20 0.37
SCN5A Q14524 1/20 0.36
HTR2A P28223 2/20 0.36
SLC6A4 P31645 1/20 0.36
DRD1 P21728 1/20 0.34
PNLIP P16233 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP3A4 P08684 2/20 0.33
TSHR P16473 1/20 0.33
EGFR P00533 2/20 0.32
ERBB2 P04626 2/20 0.32
ERBB3 P21860 2/20 0.32
ERBB4 Q15303 2/20 0.32
MRGPRX4 Q96LA9 1/20 0.32
SYK P43405 1/20 0.32
MPO P05164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30770141 0.84 SCN5A (0.36) DRD2DRD4DRD3SCN5AHTR2A
SCHEMBL26697694 0.84 SCN5A (0.36) DRD2DRD4DRD3SCN5AHTR2A
SCHEMBL3483796 0.82 PDE7A (0.41) DRD2DRD4DRD3PDE7ASCN5A
SCHEMBL29887886 0.77 EGFR (0.38) PDE7AHTR2ASLC6A4EGFRERBB2
SCHEMBL3484112 0.77 EGFR (0.38) PDE7AHTR2ASLC6A4EGFRERBB2
SCHEMBL3483989 0.74 AXL (0.41) DRD2DRD4DRD3MEN1KMT2A
SCHEMBL3484000 0.73 PDE7A (0.37) PDE7AHTR2ASLC6A4PNLIPMEN1
SCHEMBL7187883 0.73 MAOB (0.55) PDE7AHTR2ASLC6A4MEN1KMT2A
SCHEMBL3064096 0.72 SCN5A (0.42) DRD2DRD4DRD3SCN5AMEN1
SCHEMBL631854 0.71 PDE7A (0.49) PDE7AHTR2ASLC6A4PNLIPMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021231400-A1 BIS-ARYL ETHERS CONTAINING N-ACYL AZETIDINE AS EGFR/HER2 INHIBITORS ACCUTAR BIOTECHNOLOGY, INC. (US) 2021-11-18 WO disclosed
US-20100004238-A1 FUSED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-01-07 US disclosed
EP-2103620-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-09-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100004238-A1 FUSED HETEROCYCLIC COMPOUND ERBB2, ROS1, FLT3 DRD2 1841/4885DRD4 2385/4885DRD3 2397/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.