Tryptophan

Tryptophan

SCHEMBL3515219

NCCCC[C@H](N)C(=O)O.NCCCC[C@H](N)C(=O)O.N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARDPTGS1PTGS2dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Tryptophan. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.78
MAPT P10636 3/20 0.78
KMT2A Q03164 3/20 0.78
LMNA P02545 2/20 0.78
TSHR P16473 2/20 0.78
BLM P54132 2/20 0.78
PMP22 Q01453 2/20 0.78
MEN1 O00255 2/20 0.78
MPO P05164 1/20 0.78
HIF1A Q16665 1/20 0.78
MC4R P32245 2/20 0.61
MC5R P33032 1/20 0.61
MC3R P41968 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.56
APAF1 O14727 1/20 0.55
POLB P06746 1/20 0.55
RECQL P46063 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
HTR1A P08908 2/20 0.55
HTR2A P28223 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tryptophan SCHEMBL1781955 1.00 KDM4E (0.78) KDM4EMAPTKMT2ALMNATSHR
Dl-Tryptophan SCHEMBL2255452 1.00 KDM4E (0.78) KDM4EMAPTKMT2ALMNATSHR
Dl-Tryptophan SCHEMBL30058301 1.00 KDM4E (0.78) KDM4EMAPTKMT2ALMNATSHR
Dl-Tryptophan SCHEMBL26981429 1.00 KDM4E (0.78) KDM4EMAPTKMT2ALMNATSHR
Dl-Tryptophan SCHEMBL27153934 1.00 KDM4E (0.78) KDM4EMAPTKMT2ALMNATSHR
Dl-Tryptophan SCHEMBL27705509 0.96 KDM4E (0.80) KDM4EMAPTKMT2ALMNATSHR
Dl-Tryptophan SCHEMBL21219049 0.95 KMT2A (0.71) KDM4EMAPTKMT2ALMNATSHR
Tryptophan SCHEMBL6030686 0.94 KDM4E (0.70) KDM4EMAPTKMT2ALMNATSHR
Tryptophan SCHEMBL14719809 0.92 KDM4E (0.67) KDM4EMAPTKMT2ALMNATSHR
Dl-Tryptophan SCHEMBL27584251 0.92 KDM4E (0.67) KDM4EMAPTKMT2ALMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4301790-A1 SUNSCREENS DERIVED FROM KYNURENINES AND OTHER UV-ABSORBING OXIDIZED AMINO ACIDS BOUND TO PEPTIDES OR POLYMERS The Trustees Of Princeton University (US) 2024-01-10 EP disclosed
CN-116444603-A Tryptophan-containing antibacterial peptide and synthesis method and application thereof 江苏大学 2023-07-18 CN disclosed
CN-116444603-A Tryptophan-containing antibacterial peptide and synthesis method and application thereof 江苏大学 2023-07-18 CN disclosed
US-20100311821-A1 Synthetic vector UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. 2010-12-09 US disclosed
WO-1995026733-A1 OLIGONUCLEOSIDE CLEAVAGE COMPOUNDS AND THERAPIES GENTA INCORPORATED (US) 1995-10-12 WO disclosed