SCHEMBL3516443

SCHEMBL3516443

COc1ccc(-c2ccnc(Nc3ccc(S(=O)(=O)NCCCN(C)C)c(C(F)(F)F)c3)n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.51
IKBKB O14920 5/20 0.51
CNR1 P21554 3/20 0.48
PIK3CA P42336 4/20 0.47
PIK3CG P48736 4/20 0.47
PIK3CB P42338 3/20 0.47
GSK3B P49841 1/20 0.45
CDK5 Q00535 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
SYK P43405 1/20 0.44
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
CCNA1 P78396 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3520485 0.95 IKBKB (0.50) CNR2IKBKBCNR1PIK3CAPIK3CG
SCHEMBL3520096 0.89 IKBKB (0.49) CNR2IKBKBCNR1SYKCCNA2
SCHEMBL3516351 0.88 IKBKB (0.53) IKBKBPIK3CAPIK3CGPIK3CBCDK5
SCHEMBL3518027 0.88 IKBKB (0.53) IKBKBPIK3CAPIK3CGPIK3CBCDK5
SCHEMBL3521916 0.84 IKBKB (0.47) CNR2IKBKBCNR1CCNA2CDK2
SCHEMBL3518123 0.82 IKBKB (0.52) IKBKBPIK3CAPIK3CGPIK3CBCDK5
SCHEMBL3522470 0.82 PIK3CG (0.54) IKBKBPIK3CAPIK3CGPIK3CBCDK5
SCHEMBL3518567 0.82 PIK3CG (0.58) IKBKBPIK3CAPIK3CGPIK3CBGSK3B
SCHEMBL4872194 0.81 IKBKB (0.62) IKBKBCDK2
SCHEMBL3522392 0.78 IKBKB (0.70) IKBKBPIK3CAPIK3CGPIK3CBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7799915-B2 Anilino-pyrimidine analogs WYETH LLC (US) 2010-09-21 US claimed
EP-1799652-A1 N-BENZENESULFONYL SUBSTITUTED ANILINO-PYRIMIDINE ANALOGS Wyeth (US) 2007-06-27 EP claimed
WO-2006044457-A1 N-BENZENESULFONYL SUBSTITUTED ANILINO-PYRIMIDINE ANALOGS WYETH (US) 2006-04-27 WO claimed