SCHEMBL3519043

SCHEMBL3519043

Nc1ncn(CCC2CCN(C(=O)O)CC2)c2nc(Br)nc1-2

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 10/20 0.34
HSP90AB1 P08238 10/20 0.34
TGFBR1 P36897 2/20 0.34
BTK Q06187 2/20 0.33
CPB1 P15086 1/20 0.33
CPB2 Q96IY4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3124566 0.90 TGFBR1 (0.42) HSP90AA1HSP90AB1TGFBR1
SCHEMBL3750656 0.86 FAAH (0.42) TGFBR1
SCHEMBL3519511 0.83 TGFBR1 (0.39) TGFBR1BTKCPB1CPB2
SCHEMBL3116823 0.83 HSP90AA1 (0.38) HSP90AA1HSP90AB1TGFBR1
SCHEMBL3116808 0.83 HSP90AA1 (0.38) HSP90AA1HSP90AB1TGFBR1
SCHEMBL3115893 0.79 HSP90AA1 (0.52) HSP90AA1HSP90AB1
SCHEMBL3111542 0.74 ERBB2 (0.36) HSP90AA1HSP90AB1
SCHEMBL3113538 0.74 HSP90AA1 (0.49) HSP90AA1HSP90AB1
SCHEMBL3114224 0.74 HSP90AA1 (0.49) HSP90AA1HSP90AB1
SCHEMBL3114213 0.74 HSP90AA1 (0.49) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2219448-A1 THERAPEUTIC COMPOUNDS AND THEIR USE IN TREATING DISEASES AND DISORDERS Myriad Pharmaceuticals, Inc. (US) 2010-08-25 EP disclosed
WO-2009065035-A1 THERAPEUTIC COMPOUNDS AND THEIR USE IN TREATING DISEASES AND DISORDERS MYRIAD GENETICS, INC. (US) 2009-05-22 WO disclosed