SCHEMBL3528084

SCHEMBL3528084

O=C(Nc1ncc2c(n1)CCN(C(=O)c1sc3ccccc3c1Cl)C2)c1cccs1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.49
HTT P42858 2/20 0.47
ALDH1A1 P00352 6/20 0.44
LMNA P02545 2/20 0.44
KMT2A Q03164 2/20 0.42
PDGFRB P09619 4/20 0.42
KDM4E B2RXH2 5/20 0.41
NPC1 O15118 4/20 0.41
MAPT P10636 4/20 0.41
RAB9A P51151 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
HPGD P15428 2/20 0.41
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ENPP2 Q13822 1/20 0.40
MAPK1 P28482 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3533825 0.88 PDGFRB (0.50) KDRHTTALDH1A1LMNAKMT2A
SCHEMBL3529825 0.81 HSP90AB1 (0.53) KDRALDH1A1LMNAKMT2APDGFRB
SCHEMBL3529823 0.80 ALDH1A1 (0.50) ALDH1A1LMNAKMT2APDGFRBKDM4E
SCHEMBL3531360 0.73 HSP90AB1 (0.47) KDRHTTALDH1A1LMNAPDGFRB
SCHEMBL10207563 0.73 ALDH1A1 (0.48) ALDH1A1LMNAKMT2AKDM4ENPC1
SCHEMBL12204214 0.72 ALDH1A1 (0.57) HTTALDH1A1LMNAKMT2ANPC1
SCHEMBL3533372 0.69 HSP90AB1 (0.47) KDRHTTLMNAPDGFRBKDM4E
SCHEMBL3532057 0.69 LMNA (0.44) KDRHTTLMNAPDGFRBMAPT
SCHEMBL3531179 0.69 PDGFRB (0.46) KDRHTTALDH1A1LMNAPDGFRB
SCHEMBL3530952 0.68 NPC1 (0.51) KDRKMT2APDGFRBNPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7662828-B2 Substituted 5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine-2-yl compounds and 5,6,7,8-tetrahydroquinazoline-2-yl compounds GRUENENTHAL GMBH (DE) 2010-02-16 US claimed