SCHEMBL3529903

SCHEMBL3529903

NS(=O)(=O)c1c[c]c(O)c2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.56
CDK2 P24941 1/20 0.52
CYP2C9 P11712 2/20 0.46
MCL1 Q07820 2/20 0.46
HSD17B10 Q99714 1/20 0.46
CA2 P00918 8/20 0.44
CA1 P00915 7/20 0.44
CA9 Q16790 6/20 0.44
FTO Q9C0B1 1/20 0.40
CA6 P23280 4/20 0.39
CA5A P35218 4/20 0.39
CA4 P22748 3/20 0.39
CA12 O43570 3/20 0.39
CA7 P43166 3/20 0.39
CA5B Q9Y2D0 3/20 0.39
CA14 Q9ULX7 2/20 0.39
MPL P40238 1/20 0.38
HKDC1 Q2TB90 1/20 0.37
ALPL P05186 1/20 0.35
ALPI P09923 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5033149 0.83 TTR (0.43) LDHACDK2MPLHKDC1
SCHEMBL1535644 0.73 IDO1 (0.50) LDHAHSD17B10CA2CA5ACA4
SCHEMBL1805457 0.72 LDHA (1.00) LDHACDK2CYP2C9MCL1HSD17B10
SCHEMBL2325097 0.70 IDO1 (0.35)
SCHEMBL7535265 0.69 MCL1 (0.67) LDHACDK2CYP2C9MCL1HSD17B10
SCHEMBL588923 0.68 CDK2 (1.00) LDHACDK2CYP2C9MCL1HSD17B10
SCHEMBL29401806 0.68 CDK2 (1.00) LDHACDK2CYP2C9MCL1HSD17B10
SCHEMBL9138970 0.68 CDK2 (0.78) LDHACDK2CYP2C9MCL1HSD17B10
SCHEMBL6633977 0.68 TTR (0.43) LDHAMPLTDP1
SCHEMBL10605483 0.68 LDHA (0.58) LDHACDK2CYP2C9MCL1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7709479-B1 Quinazoline derivatives and their use as pharmaceuticals ASTRAZENECA (SE) 2010-05-04 US disclosed
CN-1391562-A Quinazoline derivatives as medicaments ASTRAZENECA AB (SE) 2003-01-15 CN disclosed