SCHEMBL353004

SCHEMBL353004

CNC(=O)C1CCC(=O)O1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.43
CA9 Q16790 1/20 0.43
CYP1A2 P05177 2/20 0.33
IKBKB O14920 1/20 0.31
PRKCA P17252 3/20 0.30
NFKB1 P19838 1/20 0.30
NFKB2 Q00653 1/20 0.30
RELA Q04206 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12104209 1.00 CA1 (0.43) CA1CA9CYP1A2IKBKBPRKCA
SCHEMBL15334751 1.00 CA1 (0.43) CA1CA9CYP1A2IKBKBPRKCA
SCHEMBL16804836 0.89 CA1 (0.36) CA1CA9
SCHEMBL16804841 0.89 CA1 (0.36) CA1CA9
SCHEMBL22268208 0.83 CA1 (0.39) CA1CA9
SCHEMBL19818951 0.83 CA1 (0.39) CA1CA9
SCHEMBL17323381 0.83 CA1 (0.39) CA1CA9
SCHEMBL12108375 0.79 CYP2C9 (0.41) CA1CA9CYP1A2PRKCA
SCHEMBL12108376 0.79 CYP2C9 (0.41) CA1CA9CYP1A2PRKCA
SCHEMBL12104238 0.79 TSHR (0.41) CA1CA9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160046661-A1 RAS INHIBITORS AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2016-02-18 US disclosed
US-8148380-B2 Antibacterial amide and sulfonamide substituted heterocyclic urea compounds CRESTONE, INC. (US) 2012-04-03 US disclosed
US-20120015941-A1 Antibacterial Amide and Sulfonamide Substituted Heterocyclic Urea Compounds CRESTONE, INC. (US) 2012-01-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160046661-A1 RAS INHIBITORS AND USES THEREOF KRAS, NRAS, RASGRP1 CA1 2892/4885CA9 419/4885CYP1A2 2920/4885
US-20120015941-A1 Antibacterial Amide and Sulfonamide Substituted Heterocyclic Urea Compounds NAAA, AADAC, RPSA CA1 3604/4885CA9 2039/4885CYP1A2 2181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.