SCHEMBL3553616

SCHEMBL3553616

CCc1c(C(=O)c2ccc(Cl)cc2Cl)oc2cc(-c3cccnc3)ccc12

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 6/20 0.47
MKNK2 Q9HBH9 6/20 0.47
MAPT P10636 1/20 0.41
KLK7 P49862 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
GAA P10253 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
CAPN1 P07384 1/20 0.38
CYP19A1 P11511 1/20 0.38
PIM1 P11309 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
P2RX7 Q99572 1/20 0.37
CNR1 P21554 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3562497 0.87 MKNK1 (0.49) MKNK1MKNK2MAPTKLK7CYP19A1
SCHEMBL3319291 0.85 MKNK1 (0.52) MKNK1MKNK2MAPTKLK7CAPN1
SCHEMBL3098576 0.84 MKNK1 (0.48) MKNK1MKNK2MAPTKLK7CYP1A2
Hydrochloric Acid SCHEMBL3319623 0.84 MKNK1 (0.51) MKNK1MKNK2MAPTKLK7CAPN1
SCHEMBL13335837 0.83 MKNK1 (0.45) MKNK1MKNK2MAPTKLK7CYP11B2
SCHEMBL3100585 0.82 XDH (0.39) MAPT
SCHEMBL3564020 0.81 HSD17B1 (0.43) MAPTGAACYP11B1CYP11B2CNR1
SCHEMBL13335719 0.76 MKNK1 (0.50) MKNK1MKNK2MAPTKLK7CAPN1
SCHEMBL3089232 0.76 MKNK1 (0.55) MKNK1MKNK2KLK7CYP1A2CYP2C9
SCHEMBL13335726 0.75 MKNK1 (0.48) MKNK1MKNK2MAPTCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7659412-B2 Benzofuran derivatives useful for treating hyper-proliferative disorders BAYER HEALTHCARE LLC (US) 2010-02-09 US disclosed
US-20090023783-A1 BENZOFURAN DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS ZHANG CHENGZHI 2009-01-22 US disclosed
US-7420066-B2 Benzofuran derivatives useful for treating hyper-proliferative disorders BAYER PHARMACEUTICALS CORPORATION (US) 2008-09-02 US disclosed
US-20060194816-A1 Benzofuran derivatives useful for treating hyper-proliferative disorders BAER PHAMACEUTICALS CORPORATION (US) 2006-08-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060194816-A1 Benzofuran derivatives useful for treating hyper-proliferative disorders MKI67, PCNA, CCNI MKNK1 1953/4885MKNK2 2039/4885MAPT 4163/4885
US-20090023783-A1 BENZOFURAN DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS PCNA, MKI67, CDK4 MKNK1 2068/4885MKNK2 2279/4885MAPT 4197/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.