SCHEMBL3555860

SCHEMBL3555860

N=C(N)c1cccc(F)c1F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.56
CES1 P23141 4/20 0.56
BCHE P06276 1/20 0.56
HPGD P15428 1/20 0.43
CTSL P07711 1/20 0.38
ALB P02768 1/20 0.38
BACE1 P56817 1/20 0.37
KAT6A Q92794 1/20 0.37
F2 P00734 2/20 0.36
F10 P00742 2/20 0.36
F12 P00748 1/20 0.36
F7 P08709 1/20 0.36
F3 P13726 1/20 0.36
PKM P14618 1/20 0.36
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
BLM P54132 1/20 0.34
ATM Q13315 1/20 0.34
KLK1 P06870 1/20 0.34
KLK5 Q9Y337 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3647753 0.98 CES2 (0.54) CES2CES1BCHEHPGDCTSL
Hydrochloric Acid SCHEMBL10434081 0.96 CES2 (0.52) CES2CES1BCHEHPGDCTSL
SCHEMBL29970881 0.81 CES2 (0.52) CES2CES1BCHEHPGDCTSL
SCHEMBL522903 0.81 CES2 (0.52) CES2CES1BCHEHPGDCTSL
SCHEMBL20599650 0.79 CES2 (0.54) CES2CES1BCHEF2F10
SCHEMBL16935755 0.79 CES2 (0.58) CES2CES1BCHEHPGDCTSL
Hydrochloric Acid SCHEMBL319729 0.79 CES2 (0.50) CES2CES1BCHEHPGDCTSL
SCHEMBL4223326 0.78 BACE1 (0.42) CES2CES1BCHEALBBACE1
Hydrochloric Acid SCHEMBL21553857 0.78 ALB (0.53) CES2CES1BCHEALBBACE1
SCHEMBL27971210 0.78 BACE1 (0.42) CES2CES1BACE1KAT6AF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3732183-A1 METAL COMPLEX COMPRISING AMIDINE AND THIOPHENE FUSED CYCLOPENTADIENYL LIGANDS Arlanxeo Netherlands B.V. (NL) 2020-11-04 EP disclosed
CN-107922529-A Catalyst system 阿朗新科荷兰有限公司 2018-04-17 CN disclosed
CN-107207532-A Nitroimidazole derivatives against tuberculosis 南京明德新药研发股份有限公司 2017-09-26 CN disclosed
WO-2011079118-A1 PTERIDINONES AS INHIBITORS OF POLO-LIKE KINASE ELAN PHARMACEUTICALS, INC (US) 2011-06-30 WO disclosed
US-7645776-B2 (R)-1-{2-[3-(4-Methoxy-phenyl)-[1,2,4]oxadiazol-5-yl]-piperidin-1-yl}-2-phenoxy-ethanone; carnitine-dependent palmitoyltransferases (CPTs); reduce liver beta -oxidation, consequently inhibit gluconeogenesis and therefore counteract hyperglycemia HOFFMANN-LA ROCHE INC. (US) 2010-01-12 US disclosed
CN-101622284-A Elastomeric compound DSM IP ASSETS BV 2010-01-06 CN disclosed
EP-1924611-A1 PROCESS FOR THE PREPARATION OF A METAL-ORGANIC COMPOUND COMPRISING A SPECTATOR LIGAND DSMIP Assets B.V. (NL) 2008-05-28 EP disclosed
US-20070129544-A1 (R)-1-{2-[3-(4-Methoxy-phenyl)-[1,2,4]oxadiazol-5-yl]-piperidin-1-yl}-2-phenoxy-ethanone; carnitine-dependent palmitoyltransferases (CPTs); reduce liver beta -oxidation, consequently inhibit gluconeogenesis and therefore counteract hyperglycemia F. HOFFMANN-LA ROCHE AG (CH) 2007-06-07 US disclosed
WO-2007031295-A1 PROCESS FOR THE PREPARATION OF A METAL-ORGANIC COMPOUND COMPRISING A SPECTATOR LIGAND DSM IP ASSETS B.V. (NL) 2007-03-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070129544-A1 (R)-1-{2-[3-(4-Methoxy-phenyl)-[1,2,4]oxadiazol-5-yl]-piperidin-1-yl}-2-phenoxy-ethanone; carnitine-dependent palmitoyltransferases (CPTs); reduce liver beta -oxidation, consequently inhibit gluconeogenesis and therefore counteract hyperglycemia CPT1A, CPT1B, CPT2 CES2 38/4885CES1 5/4885BCHE 1185/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.