SCHEMBL3557567

SCHEMBL3557567

O=[C]Nc1c(O)cc(O)cc1O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HPGD P15428 1/20 0.36
CES2 O00748 1/20 0.34
FASN P49327 1/20 0.34
CA12 O43570 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA7 P43166 2/20 0.33
CA9 Q16790 2/20 0.33
CA14 Q9ULX7 2/20 0.33
BACE1 P56817 1/20 0.33
TSHR P16473 1/20 0.33
GFER P55789 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK4 Q16654 1/20 0.33
NQO1 P15559 1/20 0.33
ACHE P22303 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3555814 0.81 CYP3A4 (0.48) CYP3A4HPGDALDH1A1BACE1PDK2
SCHEMBL3559875 0.80 MAOB (0.46) CYP3A4MEN1KMT2AHPGDCA12
SCHEMBL3562173 0.75 CA2 (0.39) CYP3A4HPGDCA12ALDH1A1CA1
SCHEMBL3562013 0.75 CXCR1 (0.42) MEN1KMT2ACES2CA12ALDH1A1
SCHEMBL3559775 0.72 CYP3A4 (0.48) CYP3A4MEN1KMT2ACA12CA1
SCHEMBL3555765 0.71 CYP3A4 (0.49) CYP3A4MEN1KMT2AHPGDTDP1
SCHEMBL5462195 0.70 SELL (0.42) CYP3A4MEN1KMT2AHPGDCA12
SCHEMBL5476577 0.65 CYP3A4 (0.52) CYP3A4MEN1KMT2ACA12ALDH1A1
SCHEMBL28384045 0.65 TDP1 (0.42) CYP3A4MEN1KMT2AHPGDCES2
SCHEMBL7158339 0.65 CYP3A4 (0.40) CYP3A4MEN1KMT2AHPGDCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7662826-B2 Pyrazolo [1,5-a] pyrimidine derivative and nad (p) h oxidase inhibitor containing the same SHIONOGI & CO., LTD. (JP) 2010-02-16 US disclosed
US-20060089362-A1 Pyrazolo [1,5-a] pyrimidine derivative and nad (p) h oxidase inhibitor containing the same SHIONOGI & CO., LTD (JP) 2006-04-27 US disclosed
EP-1533308-A2 A process for producing a simvastatin precursor Kaneka Corporation (JP) 2005-05-25 EP disclosed
US-6331641-B1 Process for producing simvastatin KANEKA CORPORATION (JP) 2001-12-18 US disclosed
EP-1155698-A1 ORGANOBORON COMPOUNDS EXHIBITING ANTICOCCIDIAL ACTIVITIES Nitto Kasei Co., Ltd. (JP) 2001-11-21 EP disclosed
EP-1057825-A1 ISOFLAVANE DERIVATIVES AND IMMUNOPOTENTIATING COMPOSITIONS CONTAINING THE SAME SHIONOGI & CO., LTD. (JP) 2000-12-06 EP disclosed
EP-1055671-A1 PROCESS FOR PRODUCING SIMVASTATIN KANEKA CORPORATION (JP) 2000-11-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060089362-A1 Pyrazolo [1,5-a] pyrimidine derivative and nad (p) h oxidase inhibitor containing the same NADK, PNPO, NQO1 CYP3A4 300/4885MEN1 3501/4885KMT2A 2263/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.