SCHEMBL3559265

SCHEMBL3559265

CC(C)(C)OC(=O)N(C/C=C/Cl)c1ccc2ccc(C#N)cc2c1Br

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 2/20 0.39
CCNC P24863 2/20 0.31
CDK8 P49336 2/20 0.31
CETP P11597 1/20 0.31
SCN9A Q15858 1/20 0.31
FNTA P49354 1/20 0.30
FNTB P49356 1/20 0.30
CCR9 P51686 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3559269 1.00 NCEH1 (0.39) NCEH1CCNCCDK8CETPSCN9A
SCHEMBL3564221 0.93 NCEH1 (0.47) NCEH1CETPSCN9AFNTAFNTB
SCHEMBL3564217 0.93 NCEH1 (0.47) NCEH1CETPSCN9AFNTAFNTB
SCHEMBL3846549 0.84 ALDH1A1 (0.32)
SCHEMBL3913701 0.84 ALDH1A1 (0.32)
SCHEMBL3851116 0.83 SMN1; SMN2 (0.40) NCEH1
SCHEMBL2400850 0.83 SMN1; SMN2 (0.40) NCEH1
SCHEMBL3566612 0.82 NQO2 (0.35)
SCHEMBL3562270 0.82 NQO2 (0.35)
SCHEMBL3562268 0.82 NQO2 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7718688-B2 Nitrobenzindoles and their use in cancer therapy AUCKLAND UNISERVICES LIMITED (NZ) 2010-05-18 US disclosed
EP-1809603-A4 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY AUCKLAND UNISERVICES LTD (NZ) 2009-09-02 EP disclosed
US-20080119442-A1 as hypoxia-selective drugs and radiosensitizers for cancer therapy; nitroreductase inhibitor; 1-(Chloromethyl)-5,6-dinitro-3-(5,6,7-trimethoxyindol-2-carbonyl)-1,2-dihydro-3H-benzo[e]indole; halogenation of naphthalene derivative followed by hydration and cyclization AUCKLAND UNISERVICES LIMITED (NZ) 2008-05-22 US disclosed
EP-1809603-A1 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY Auckland Uniservices Limited (NZ) 2007-07-25 EP disclosed
WO-2006043839-A1 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY AUCKLAND UNISERVICES LIMITED (NZ) 2006-04-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080119442-A1 as hypoxia-selective drugs and radiosensitizers for cancer therapy; nitroreductase inhibitor; 1-(Chloromethyl)-5,6-dinitro-3-(5,6,7-trimethoxyindol-2-carbonyl)-1,2-dihydro-3H-benzo[e]indole; halogenation of naphthalene derivative followed by hydration and cyclization HIF1AN, HYOU1, HIF1A NCEH1 479/4885CCNC 1413/4885CDK8 1300/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.