SCHEMBL3565158

SCHEMBL3565158

CN1C(=O)/C(=C\Nc2ccc(Cl)cc2)c2ccccc2C1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.44
APP P05067 3/20 0.42
KMT2A Q03164 5/20 0.41
MEN1 O00255 4/20 0.41
MAPT P10636 7/20 0.40
ALDH1A1 P00352 6/20 0.40
KDM4E B2RXH2 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 1/20 0.40
ERBB2 P04626 1/20 0.39
TSHR P16473 1/20 0.38
HPGD P15428 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
CES1 P23141 1/20 0.38
POLB P06746 3/20 0.38
LMNA P02545 2/20 0.38
APEX1 P27695 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3565159 1.00 CASP3 (0.44) CASP3APPKMT2AMEN1MAPT
SCHEMBL3563637 0.88 APP (0.50) CASP3APPMAPTALDH1A1KDM4E
SCHEMBL3563633 0.88 APP (0.50) CASP3APPMAPTALDH1A1KDM4E
SCHEMBL3576527 0.80 MEN1 (0.57) CASP3KMT2AMEN1ALDH1A1KDM4E
SCHEMBL3576525 0.80 MEN1 (0.57) CASP3KMT2AMEN1ALDH1A1KDM4E
SCHEMBL3566377 0.79 KDM4E (0.44) ALDH1A1KDM4ESMN1; SMN2
SCHEMBL3566379 0.79 KDM4E (0.44) ALDH1A1KDM4ESMN1; SMN2
SCHEMBL3573931 0.77 PPOX (0.46) CASP3KMT2AMEN1MAPTALDH1A1
SCHEMBL3573929 0.77 PPOX (0.46) CASP3KMT2AMEN1MAPTALDH1A1
SCHEMBL3565087 0.75 CASP3 (0.45) CASP3APPKMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7713994-B2 Substituted isoquinoline-1,3(2H,4H)-diones, 1-thioxo,1,4-dihydro-2H-isoquinoline-3-ones and 1,4-dihyro-3 (2H)-isoquinolones and methods of use thereof WYETH LLC (US) 2010-05-11 US claimed