SCHEMBL3570500

SCHEMBL3570500

CN1CCN(N(C(N)=O)c2ccc(NC=C3C(=O)NC(=O)c4ccc(Br)cc43)cc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.36
CCND1 P24385 1/20 0.36
CDK2 P24941 1/20 0.36
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
DUSP3 P51452 1/20 0.32
PTPN5 P54829 1/20 0.32
PTPN11 Q06124 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
CCNB2 O95067 3/20 0.32
CDK1 P06493 3/20 0.32
CCNB1 P14635 3/20 0.32
CCNB3 Q8WWL7 3/20 0.32
KMT2A Q03164 1/20 0.31
HSP90AA1 P07900 2/20 0.31
CSF1R P07333 1/20 0.31
CCR6 P51684 1/20 0.31
APP P05067 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3570497 1.00 CDK4 (0.36) CDK4CCND1CDK2KDM4EALDH1A1
SCHEMBL3561137 0.87 CSF1R (0.40) MAPTCSF1R
SCHEMBL3561141 0.87 CSF1R (0.40) MAPTCSF1R
SCHEMBL3560367 0.81 ALDH1A1 (0.44) CDK4CCND1CDK2KDM4EALDH1A1
SCHEMBL3560371 0.81 ALDH1A1 (0.44) CDK4CCND1CDK2KDM4EALDH1A1
SCHEMBL3562396 0.80 PDGFRB (0.44) CDK4CCND1CDK2ALDH1A1MAPT
SCHEMBL3562399 0.80 PDGFRB (0.44) CDK4CCND1CDK2ALDH1A1MAPT
SCHEMBL3570607 0.79 CDK4 (0.39) CDK4CCND1CDK2LMNAMAPT
SCHEMBL13344041 0.79 CDK4 (0.39) CDK4CCND1CDK2LMNAMAPT
SCHEMBL3570604 0.79 CDK4 (0.39) CDK4CCND1CDK2LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7713994-B2 Substituted isoquinoline-1,3(2H,4H)-diones, 1-thioxo,1,4-dihydro-2H-isoquinoline-3-ones and 1,4-dihyro-3 (2H)-isoquinolones and methods of use thereof WYETH LLC (US) 2010-05-11 US claimed