SCHEMBL3574435

SCHEMBL3574435

CCCCN1CCN(c2ccc(-c3nc4c(C(N)=O)cccc4[nH]3)cc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 5/20 1.00
AURKA O14965 3/20 1.00
PARP1 P09874 15/20 0.64
DHODH Q02127 2/20 0.58
PARP2 Q9UGN5 3/20 0.57
KDR P35968 3/20 0.55
PRKD3 O94806 1/20 0.55
PIM1 P11309 1/20 0.55
SRC P12931 1/20 0.55
FLT4 P35916 1/20 0.55
CLK2 P49760 1/20 0.55
GSK3A P49840 1/20 0.55
DYRK1A Q13627 1/20 0.55
PIM3 Q86V86 1/20 0.55
PRKD2 Q9BZL6 1/20 0.55
CLK4 Q9HAZ1 1/20 0.55
MKNK2 Q9HBH9 1/20 0.55
STK17A Q9UEE5 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3582845 0.96 AURKB (0.93) AURKBAURKAPARP1DHODHPARP2
SCHEMBL3582276 0.90 AURKB (0.82) AURKBAURKAPARP1DHODHPARP2
SCHEMBL3587286 0.87 AURKA (0.76) AURKBAURKAPARP1DHODHPARP2
SCHEMBL3582843 0.86 AURKB (0.76) AURKBAURKAPARP1DHODHPARP2
Hydrochloric Acid SCHEMBL6805711 0.86 AURKB (0.98) AURKBAURKAPARP1DHODHPARP2
SCHEMBL6580984 0.86 AURKB (0.75) AURKBAURKAPARP1DHODHPRKD3
SCHEMBL3574441 0.85 AURKA (0.75) AURKBAURKAPARP1
SCHEMBL6804561 0.84 AURKB (0.93) AURKBAURKAPARP1DHODHPARP2
SCHEMBL3580117 0.83 AURKB (0.77) AURKBAURKAPARP1DHODHKDR
SCHEMBL3577220 0.83 AURKA (0.71) AURKBAURKAPARP1DHODHPARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed