SCHEMBL3574441

SCHEMBL3574441

CCCCN1CCN(c2ccc(-c3nc4cccc(C(N)=O)c4[nH]3)cc2)CC1

nearest known ligand 0.75

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.75
AURKB Q96GD4 2/20 0.75
ACHE P22303 1/20 0.50
DRD2 P14416 4/20 0.48
DRD3 P35462 4/20 0.48
CHEK2 O96017 5/20 0.46
PARP1 P09874 2/20 0.46
HTR1A P08908 1/20 0.44
MT-CO2 P00403 1/20 0.43
ADORA2B P29275 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3582854 0.96 AURKB (0.70) AURKAAURKBACHEDRD2DRD3
SCHEMBL3582282 0.91 AURKB (0.61) AURKAAURKBACHEDRD2DRD3
SCHEMBL3587289 0.88 AURKA (0.56) AURKAAURKBCHEK2PARP1
SCHEMBL3582849 0.87 AURKB (0.58) AURKAAURKBACHEDRD2DRD3
SCHEMBL3574435 0.85 AURKB (1.00) AURKAAURKBPARP1
SCHEMBL3580122 0.84 AURKB (0.56) AURKAAURKBACHECHEK2PARP1
SCHEMBL3577227 0.84 AURKA (0.53) AURKAAURKBCHEK2PARP1
SCHEMBL6804570 0.84 AURKA (0.72) AURKAAURKBDRD2DRD3CHEK2
SCHEMBL3576982 0.83 AURKA (0.52) AURKAAURKBACHECHEK2PARP1
SCHEMBL6029840 0.82 AURKA (0.64) AURKAAURKBDRD2DRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed