SCHEMBL357503

SCHEMBL357503

C=C(C)N(Cc1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.47
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
CA12 O43570 2/20 0.42
CA9 Q16790 1/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
CTSL P07711 2/20 0.42
CTSB P07858 2/20 0.42
CTSS P25774 2/20 0.42
LMNA P02545 1/20 0.41
RIPK1 Q13546 2/20 0.41
MEN1 O00255 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
HTR2C P28335 1/20 0.40
SLC6A4 P31645 1/20 0.40
CA1 P00915 1/20 0.40
CA7 P43166 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3819098 0.89 AKT1 (0.52) AKT1HDAC3HDAC1HDAC2NCOR2
SCHEMBL20341352 0.88 AKT1 (0.49) AKT1HDAC3HDAC1HDAC2NCOR2
SCHEMBL22361797 0.82 AKT1 (0.50) AKT1HDAC3HDAC1HDAC2NCOR2
SCHEMBL2641206 0.80 ALDH1A1 (0.56) CA12CA9L3MBTL1LMNAMEN1
SCHEMBL22931837 0.79 KMT2A (0.58) AKT1HDAC3HDAC1HDAC2NCOR2
SCHEMBL8199047 0.79 HDAC3 (0.49) AKT1HDAC3HDAC1HDAC2NCOR2
SCHEMBL10423913 0.79 AKT1 (0.42) AKT1HDAC3HDAC1HDAC2NCOR2
SCHEMBL12003065 0.79 TSHR (0.49) HDAC1CA12CA9L3MBTL1LMNA
SCHEMBL28274515 0.79 CA12 (0.52) CA12CA9LMNARIPK1MEN1
SCHEMBL19803885 0.78 TSHR (0.50) CA12CA9LMNACA1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 253 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2104715-B1 METHOD FOR PRODUCING A WATER SELF DISPERSIBLE METALLIC OXIDE AND HYDROXIDE POWDER, POWDER AND USES THEREOF COATEX SAS (FR) 2019-03-20 EP claimed
EP-2976392-B1 USE OF A POLYMERIC EMULSION FOR THE SURFACE TREATMENT OF THE PARTICLES OF AN INORGANIC MATERIAL COATEX SAS (FR) 2018-04-25 EP claimed
EP-2222920-B1 METHOD FOR MANUFACTURING A COATING SLIP INCLUDING THE USE OF AN ACRYLIC THICKENER WITH A WATER RESISTANT CHAIN AND SLIP OBTAINED OMYA INT AG (CH) 2018-02-07 EP claimed
EP-2108007-B1 USE OF A RHEOLOGIC ADDITIVE IN THE VIBRO-COMPACTION PRODUCTION OF A FORMULATION CONTAINING WATER AND A HYDRAULIC BINDER, AND FORMULATION THUS OBTAINED COATEX SAS (FR) 2016-04-13 EP claimed
EP-2976392-A1 USE OF A POLYMERIC EMULSION FOR THE SURFACE TREATMENT OF THE PARTICLES OF AN INORGANIC MATERIAL COATEX (FR) 2016-01-27 EP claimed
EP-2129468-B1 USE AS RHEOLOGICAL AGENT IN CHARGED PLASTIC PASTE, OF DRY-GROUND CALCIUM CARBONATE WITH (METH)ACRYLIC ACID COPOLYMER WITH ALKOXY OR HYDROXY POLYALKYLENE GLYCOL FUNCTION COATEX SAS (FR) 2015-12-09 EP claimed
WO-2014147321-A1 USE OF A POLYMERIC EMULSION FOR THE SURFACE TREATMENT OF THE PARTICLES OF AN INORGANIC MATERIAL COATEX (FR) 2014-09-25 WO claimed
US-8637579-B2 Process to thicken aqueous compositions by means of organophosphate polymers COATEX S.A.S. (FR) 2014-01-28 US claimed
EP-2125235-B1 USE IN HYDRAULIC BINDER COMPOSITION OF DRY-GROUND CALCIUM CARBONATE WITH (METH)ACRYLIC ACID COPOLYMER AND ALKOXY OR HYDROXY POLYALKYLENE GLYCOL FUNCTION COATEX SAS (FR) 2013-11-27 EP claimed
EP-2379649-B1 PROCESS TO PREPARE SELF-BINDING PIGMENT PARTICLES IMPLEMENTING ACRYLIC COMB COPOLYMERS WITH HYDROPHOBIC GROUPS AS COUPLING AGENTS, SELF BINDING PIGMENT PARTICLES AND USES THEREOF OMYA INT AG (CH) 2013-11-13 EP claimed
EP-1708803-A2 USE OF STRUCTURED WATER-SOLUBLE POLYMERS OBTAINED BY CONTROLLED RADICAL POLYMERIZATION AS A DISPERSANT AND AGENT FOR ASSISTING IN THE GRINDING OF MINERAL MATERIALS COATEX S.A.S. (FR) 2006-10-11 EP claimed
US-20060162884-A1 Novel inorganic pigment containing calcium carbonate, aqueous suspension containing same, and uses thereof OMYA INTERNATIONAL AG (CH) 2006-07-27 US claimed
US-20060142498-A1 gloss activator for sheet of paper, irrespective of viewing angle; paper coating; weakly ionic water soluble acrylic-polyether (or silyloxyether) graft addition-condensation copolymer OMYA INTERNATIONAL AG (CH) 2006-06-29 US claimed
WO-2006048539-A1 SUBSTITUTED CUMYL PHENOLS, USE THEREOF IN A COPOLYMERISATION METHOD COPOLYMERS THUS OBTAINED AND USE THEREOF AS THICKENERS COATEX S.A.S. (FR) 2006-05-11 WO claimed
US-20060009560-A1 Aqueous suspensions of ground mineral materials, with low ion load and their uses OMYA INTERNATIONAL AG (CH) 2006-01-12 US claimed
EP-1572764-A1 AQUEOUS SUSPENSIONS OF GROUND MINERAL MATERIALS, WITH LOW ION LOAD AND THEIR USES Omya AG (CH) 2005-09-14 EP claimed
EP-1565504-A1 USE OF A COPOLYMER HAVING AT LEAST ONE GRAFTED ALKOXY OR HYDROXY POLYALKYLENE GLYCOL FUNCTION AS AN AGENT FOR IMPROVING OPTICAL BRIGHTENING ACTIVATION, AND PRODUCTS OBTAINED COATEX S.A.S. (FR) 2005-08-24 EP claimed
WO-2005063371-A2 USE OF STRUCTURED WATER-SOLUBLE POLYMERS OBTAINED BY CONTROLLED RADICAL POLYMERIZATION AS A DISPERSANT AND AGENT FOR ASSISTING IN THE GRINDING OF MINERAL MATERIALS COATEX S.A.S. (FR) 2005-07-14 WO claimed
WO-2004044022-A1 USE OF A COPOLYMER HAVING AT LEAST ONE GRAFTED ALKOXY OR HYDROXY POLYALKYLENE GLYCOL FUNCTION AS AN AGENT FOR IMPROVING OPTICAL BRIGHTENING ACTIVATION, AND PRODUCTS OBTAINED COATEX S.A.S. (FR) 2004-05-27 WO claimed
WO-2004041882-A1 AQUEOUS SUSPENSIONS OF GROUND MINERAL MATERIALS, WITH LOW ION LOAD AND THEIR USES OMYA AG (CH) 2004-05-21 WO claimed