SCHEMBL3575162

SCHEMBL3575162

CCOC(=O)c1cccc2[nH]c(-c3ccc(N4CCN(C)CC4)cc3)nc12

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 3/20 0.72
PRKD3 O94806 1/20 0.72
MAP4K4 O95819 1/20 0.72
PIM1 P11309 1/20 0.72
CLK2 P49760 1/20 0.72
MAP4K2 Q12851 1/20 0.72
CAMK2D Q13557 1/20 0.72
DYRK1A Q13627 1/20 0.72
PIM3 Q86V86 1/20 0.72
PRKD2 Q9BZL6 1/20 0.72
CLK4 Q9HAZ1 1/20 0.72
STK17A Q9UEE5 1/20 0.72
MAP4K5 Q9Y4K4 1/20 0.72
AURKA O14965 2/20 0.62
PARP1 P09874 11/20 0.59
SIRT2 Q8IXJ6 2/20 0.52
SIRT1 Q96EB6 2/20 0.52
PARP2 Q9UGN5 4/20 0.52
PKN1 Q16512 1/20 0.49
PKN2 Q16513 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3587286 0.84 AURKA (0.76) AURKBAURKAPARP1PARP2PLA2G2A
SCHEMBL3575168 0.84 SIRT2 (0.52) AURKBPRKD3MAP4K4PIM1CLK2
SCHEMBL3581187 0.84 AURKB (0.64) AURKBPRKD3MAP4K4PIM1CLK2
SCHEMBL6948231 0.81 PARP1 (0.69) AURKBPRKD3MAP4K4PIM1CLK2
SCHEMBL3577220 0.81 AURKA (0.71) AURKBAURKAPARP1PARP2PLA2G2A
SCHEMBL6810422 0.80 PKN1 (0.76) AURKBPRKD3MAP4K4PIM1CLK2
SCHEMBL7822007 0.79 MGAM (0.59) AURKBAURKAPARP1ALDH1A1SMN1; SMN2
SCHEMBL3577852 0.79 AURKB (0.61) AURKBPRKD3MAP4K4PIM1CLK2
SCHEMBL3582276 0.78 AURKB (0.82) AURKBAURKAPARP1PARP2PLA2G2A
SCHEMBL6581295 0.78 AURKB (0.56) AURKBPRKD3MAP4K4PIM1CLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed