SCHEMBL3577852

SCHEMBL3577852

CCOC(=O)c1cccc2[nH]c(-c3ccc(-n4ccnc4)cc3)nc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 5/20 0.61
MAP4K4 O95819 3/20 0.61
PIM1 P11309 3/20 0.61
CLK2 P49760 3/20 0.61
DYRK1A Q13627 3/20 0.61
PIM3 Q86V86 3/20 0.61
PRKD2 Q9BZL6 3/20 0.61
CLK4 Q9HAZ1 3/20 0.61
STK17A Q9UEE5 3/20 0.61
PRKD3 O94806 2/20 0.61
CAMK2D Q13557 2/20 0.61
MAP4K2 Q12851 2/20 0.61
MAP4K5 Q9Y4K4 2/20 0.61
PARP1 P09874 7/20 0.58
PKN1 Q16512 4/20 0.53
PKN2 Q16513 4/20 0.53
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
MITF O75030 1/20 0.50
ALDH1A1 P00352 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583754 0.85 KDM4E (0.47) AURKBMAP4K4PIM1CLK2DYRK1A
SCHEMBL3577856 0.84 KDM4E (0.50) AURKBMAP4K4PIM1CLK2DYRK1A
SCHEMBL3575386 0.83 PARP1 (0.67) AURKBMAP4K4PIM1CLK2DYRK1A
SCHEMBL6810422 0.83 PKN1 (0.76) AURKBMAP4K4PIM1CLK2DYRK1A
SCHEMBL3585590 0.83 PKN1 (0.54) AURKBMAP4K4PIM1CLK2DYRK1A
SCHEMBL6948231 0.81 PARP1 (0.69) AURKBMAP4K4PIM1CLK2DYRK1A
SCHEMBL3575162 0.79 AURKB (0.72) AURKBMAP4K4PIM1CLK2DYRK1A
SCHEMBL7480831 0.78 PKN1 (0.67) AURKBMAP4K4PIM1CLK2DYRK1A
SCHEMBL6578697 0.77 HPSE (0.47) AURKBMAP4K4PIM1CLK2DYRK1A
SCHEMBL3580402 0.76 PARP1 (0.69) AURKBMAP4K4PIM1CLK2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed