SCHEMBL3576336

SCHEMBL3576336

CC(C)(C)OC(=O)N1CCCN(c2ccc(-c3nc4c(C(N)=O)cccc4[nH]3)cc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.62
AURKA O14965 1/20 0.60
AURKB Q96GD4 1/20 0.60
DHODH Q02127 3/20 0.57
PARP2 Q9UGN5 2/20 0.54
PLA2G2A P14555 1/20 0.52
ALOX15 P16050 1/20 0.52
PTGS2 P35354 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6578514 0.88 ATR (0.51) PARP1AURKAAURKBDHODHPARP2
SCHEMBL3576337 0.86 PARP1 (0.49) PARP1AURKAAURKB
SCHEMBL31413289 0.85 PARP1 (0.72) PARP1DHODHPLA2G2AALOX15PTGS2
SCHEMBL3574580 0.83 AURKA (0.66) PARP1AURKAAURKBDHODHPARP2
SCHEMBL3577220 0.83 AURKA (0.71) PARP1AURKAAURKBDHODHPARP2
SCHEMBL16107567 0.82 PARP1 (0.73) PARP1PARP2
SCHEMBL3587286 0.81 AURKA (0.76) PARP1AURKAAURKBDHODHPARP2
SCHEMBL3582843 0.81 AURKB (0.76) PARP1AURKAAURKBDHODHPARP2
SCHEMBL3579915 0.81 PARP1 (0.67) PARP1AURKAAURKBDHODHPARP2
SCHEMBL3582368 0.78 AURKB (0.64) PARP1AURKAAURKBDHODHPARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed