SCHEMBL3576337

SCHEMBL3576337

CC(C)(C)OC(=O)N1CCCN(c2ccc(-c3nc4cccc(C(N)=O)c4[nH]3)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.49
ATR Q13535 1/20 0.47
AURKA O14965 1/20 0.45
AURKB Q96GD4 1/20 0.45
CHEK2 O96017 9/20 0.45
CKS1B P61024 1/20 0.44
SKP1 P63208 1/20 0.44
SKP2 Q13309 1/20 0.44
GPR119 Q8TDV5 1/20 0.43
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
JAK2 O60674 1/20 0.42
JAK3 P52333 1/20 0.42
PRMT5 O14744 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3576336 0.86 PARP1 (0.62) PARP1AURKAAURKB
SCHEMBL3574583 0.83 AURKB (0.49) PARP1AURKAAURKBCHEK2
SCHEMBL3577227 0.83 AURKA (0.53) PARP1AURKAAURKBCHEK2ALDH1A1
SCHEMBL3587289 0.81 AURKA (0.56) PARP1AURKAAURKBCHEK2ALDH1A1
SCHEMBL3579920 0.81 AURKA (0.49) PARP1AURKAAURKBCHEK2
SCHEMBL3582849 0.81 AURKB (0.58) PARP1AURKAAURKBCHEK2
SCHEMBL3582854 0.79 AURKB (0.70) PARP1AURKAAURKBCHEK2
SCHEMBL3582373 0.78 PARP1 (0.49) PARP1ATRAURKAAURKBCHEK2
SCHEMBL3576982 0.78 AURKA (0.52) PARP1AURKAAURKBCHEK2
SCHEMBL3582282 0.78 AURKB (0.61) PARP1AURKAAURKBCHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed