SCHEMBL3582368

SCHEMBL3582368

NC(=O)c1cccc2[nH]c(-c3ccc(N4CCCNCC4)cc3)nc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 2/20 0.64
AURKA O14965 1/20 0.64
PARP1 P09874 18/20 0.62
PARP2 Q9UGN5 5/20 0.61
DHODH Q02127 2/20 0.60
PLK4 O00444 1/20 0.57
MAPK13 O15264 1/20 0.57
DYRK3 O43781 1/20 0.57
ROCK2 O75116 1/20 0.57
RPS6KA5 O75582 1/20 0.57
PRKD3 O94806 1/20 0.57
MAP4K4 O95819 1/20 0.57
CHEK2 O96017 1/20 0.57
PIM1 P11309 1/20 0.57
PHKG2 P15735 1/20 0.57
PRKACA P17612 1/20 0.57
RPS6KB1 P23443 1/20 0.57
CSNK1D P48730 1/20 0.57
CLK2 P49760 1/20 0.57
GSK3A P49840 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580352 0.96 AURKB (0.68) AURKBAURKAPARP1PARP2DHODH
SCHEMBL6812389 0.86 AURKA (0.67) AURKBAURKAPARP1PARP2DHODH
SCHEMBL3582857 0.85 PARP1 (0.66) AURKBPARP1PARP2DHODHPLK4
SCHEMBL6581733 0.85 PARP1 (0.56) AURKBAURKAPARP1PARP2DHODH
SCHEMBL3577220 0.84 AURKA (0.71) AURKBAURKAPARP1PARP2DHODH
SCHEMBL3587286 0.84 AURKA (0.76) AURKBAURKAPARP1PARP2DHODH
SCHEMBL3582373 0.83 PARP1 (0.49) AURKBAURKAPARP1PARP2CHEK2
SCHEMBL5621907 0.82 PARP1 (0.66) PARP1
SCHEMBL3579915 0.82 PARP1 (0.67) AURKBAURKAPARP1PARP2DHODH
SCHEMBL3582843 0.82 AURKB (0.76) AURKBAURKAPARP1PARP2DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed