SCHEMBL3577375

SCHEMBL3577375

CN(C)CCNc1n[c]no1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.35
DNM2 P50570 10/20 0.34
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34
CSNK2A1 P68400 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
PRMT3 O60678 1/20 0.32
CARM1 Q86X55 1/20 0.32
PRMT6 Q96LA8 1/20 0.32
PRMT1 Q99873 1/20 0.32
PRMT8 Q9NR22 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HRH4 Q9H3N8 1/20 0.30
GAA P10253 1/20 0.30
ALPG P10696 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13116703 0.67 HSD17B10 (0.38) CYP2C19DNM2CSNK2A2CSNK2BCSNK2A1
SCHEMBL932573 0.62 CYP2C19 (0.53) CYP2C19DNM2HRH3HRH4GAA
SCHEMBL18239960 0.62 DNM2 (0.47) CYP2C19DNM2HRH3
SCHEMBL11378396 0.59 ALDH1A1 (0.49) CYP2C19DNM2HRH3HRH4GAA
SCHEMBL933805 0.58 CYP2C19 (0.44) CYP2C19DNM2HRH3HRH4GAA
SCHEMBL3561186 0.57
SCHEMBL5596454 0.57 CYP2C19 (0.44) CYP2C19DNM2HRH3HRH4GAA
SCHEMBL3058517 0.57 POLB (0.58) CSNK2A2CSNK2BCSNK2A1HRH3HSD17B10
SCHEMBL24831580 0.56 DNM2 (0.43) DNM2PRMT3CARM1PRMT6PRMT1
SCHEMBL5622381 0.56 ALDH1A1 (0.62) CYP2C19DNM2HRH3HRH4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7812165-B2 6-substituted pyridoindolone derivatives, production and therapeutic use thereof SANOFI-AVENTIS (FR) 2010-10-12 US claimed
EP-1742947-B1 6-SUBSTITUTED PYRIDOINDOLONE DERIVATIVES PRODUCTION AND THERAPEUTIC USE THEREOF SANOFI AVENTIS (FR) 2008-08-20 EP claimed
US-20070129365-A1 6-Substituted pyridoindolone derivatives, production and therapeutic use thereof SANOFI-AVENTIS (FR) 2007-06-07 US claimed
US-7812165-B2 6-substituted pyridoindolone derivatives, production and therapeutic use thereof SANOFI-AVENTIS (FR) 2010-10-12 US disclosed
US-20070129365-A1 6-Substituted pyridoindolone derivatives, production and therapeutic use thereof SANOFI-AVENTIS (FR) 2007-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070129365-A1 6-Substituted pyridoindolone derivatives, production and therapeutic use thereof PNPO, CYP2D6, DPYD CYP2C19 72/4885DNM2 3298/4885CSNK2A2 3741/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.