SCHEMBL3581175

SCHEMBL3581175

CNc1ncc(Cl)cc1C(=O)N(CCc1ccnc(Cl)c1)Cc1ccc(C(C)(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 2/20 0.36
CCR9 P51686 4/20 0.36
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
C5AR1 P21730 1/20 0.33
ESRRB O95718 1/20 0.33
CNR1 P21554 1/20 0.33
F10 P00742 3/20 0.32
HSP90AA1 P07900 1/20 0.32
TP53 P04637 2/20 0.32
MAPT P10636 1/20 0.32
PIK3C3 Q8NEB9 1/20 0.32
NR1H4 Q96RI1 1/20 0.32
KLKB1 P03952 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3576692 0.89 ESRRG (0.37) ESRRGCCR9C5AR1ESRRBCNR1
SCHEMBL3581193 0.87 CCR9 (0.39) CCR9C5AR1F10KLKB1
SCHEMBL3570653 0.85 CNR1 (0.39) C5AR1CNR1HDAC8HDAC6
SCHEMBL3582723 0.84 HCRTR1 (0.37) ESRRGCCR9HCRTR1HCRTR2F10
SCHEMBL3576379 0.84 HSP90AA1 (0.46) CCR9HSP90AA1HDAC3HDAC8HDAC6
SCHEMBL3577915 0.81 F10 (0.38) ESRRGCCR9CNR1F10TP53
SCHEMBL3580374 0.81 ESRRG (0.36) ESRRGCCR9ESRRBHSP90AA1TP53
SCHEMBL3569329 0.81 C5AR1 (0.41) C5AR1CNR1F10KLKB1
SCHEMBL1397638 0.81 HCRTR1 (0.37) CCR9HCRTR1HCRTR2
SCHEMBL3587153 0.80 ESRRG (0.36) ESRRGHCRTR1HCRTR2C5AR1ESRRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed