SCHEMBL3576379

SCHEMBL3576379

CCCCN(Cc1ccc(C(C)(C)C)cc1)C(=O)c1cc(Cl)cnc1NC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.46
LTB4R2 Q9NPC1 2/20 0.41
HDAC1 Q13547 8/20 0.41
HDAC6 Q9UBN7 8/20 0.41
HDAC3 O15379 4/20 0.41
HDAC2 Q92769 4/20 0.41
HDAC4 P56524 2/20 0.41
HDAC7 Q8WUI4 2/20 0.41
HDAC10 Q969S8 2/20 0.41
HDAC11 Q96DB2 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC9 Q9UKV0 2/20 0.41
HDAC5 Q9UQL6 2/20 0.41
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CCR9 P51686 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
CNR2 P34972 1/20 0.37
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3576692 0.86 ESRRG (0.37) HSP90AA1CCR9
SCHEMBL3577915 0.85 F10 (0.38) CCR9
SCHEMBL3581175 0.84 ESRRG (0.36) HSP90AA1HDAC6HDAC3HDAC8CCR9
SCHEMBL3570653 0.82 CNR1 (0.39) HDAC1HDAC6HDAC11HDAC8CYP2D6
SCHEMBL3582723 0.81 HCRTR1 (0.37) CCR9
SCHEMBL3580812 0.80 TRPM8 (0.35) HSP90AA1HDAC6HDAC3HDAC8CCR9
SCHEMBL3584236 0.80 HCRTR1 (0.42)
SCHEMBL3569329 0.79 C5AR1 (0.41)
SCHEMBL3574298 0.79 KDM4E (0.36) CCR9
SCHEMBL3587153 0.79 ESRRG (0.36) HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed