SCHEMBL358670

SCHEMBL358670

Cc1c2cccc(C(N)=O)c2nn1C1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.52
GPR119 Q8TDV5 3/20 0.43
NR3C1 P04150 2/20 0.42
TP53 P04637 1/20 0.41
PRKCG P05129 1/20 0.41
PRKCB P05771 1/20 0.41
PRKCA P17252 1/20 0.41
PRKCH P24723 1/20 0.41
PRKCE Q02156 1/20 0.41
PRKCD Q05655 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL368905 0.96 PARP1 (0.49) PARP1GPR119NR3C1
SCHEMBL358653 0.94 PARP1 (0.47) PARP1GPR119NR3C1
SCHEMBL360298 0.91 PARP1 (0.47) PARP1
SCHEMBL358681 0.90 EED (0.46) PARP1GPR119NR3C1PRKCGPRKCB
SCHEMBL359239 0.89 PARP1 (0.51) PARP1GPR119NR3C1
SCHEMBL359678 0.89 PARP1 (0.47) PARP1
SCHEMBL359223 0.87 PARP1 (0.49) PARP1GPR119
SCHEMBL10173016 0.85 PARP1 (0.51) PARP1
SCHEMBL359388 0.83 PARP1 (0.50) PARP1
SCHEMBL370739 0.82 PARP1 (0.46) PARP1GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed