SCHEMBL359388

SCHEMBL359388

CC(C)(C)OC(=O)N1CCC(n2nc3c(C(N)=O)cccc3c2Br)C1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.50
BTK Q06187 1/20 0.43
JAK2 O60674 3/20 0.42
JAK1 P23458 3/20 0.42
SRC P12931 3/20 0.42
EGFR P00533 2/20 0.42
ABL1 P00519 1/20 0.42
ABL2 P42684 1/20 0.42
PIK3CD O00329 1/20 0.40
PIK3R2 O00459 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PIK3CG P48736 1/20 0.40
PIK3R5 Q8WYR1 1/20 0.40
PIK3R3 Q92569 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL359451 0.94 PARP1 (0.51) PARP1BTKJAK2JAK1PIK3CD
SCHEMBL359239 0.94 PARP1 (0.51) PARP1
SCHEMBL358920 0.83 NR3C1 (0.43) PARP1
SCHEMBL358670 0.83 PARP1 (0.52) PARP1
SCHEMBL360298 0.81 PARP1 (0.47) PARP1JAK2JAK1
SCHEMBL359223 0.81 PARP1 (0.49) PARP1BTKJAK2JAK1SRC
SCHEMBL357915 0.81 PARP1 (0.43) PARP1
SCHEMBL361173 0.80 PARP1 (0.41) PARP1
SCHEMBL368905 0.80 PARP1 (0.49) PARP1
SCHEMBL359678 0.79 PARP1 (0.47) PARP1JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed