SCHEMBL3589372

SCHEMBL3589372

CCOC(=O)c1cccc2nc(-c3cccc(OCCN(CC)CC)c3)[nH]c12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.55
ADORA1 P30542 2/20 0.55
MAP4K4 O95819 2/20 0.48
PIM1 P11309 2/20 0.48
PIM3 Q86V86 2/20 0.48
AURKB Q96GD4 2/20 0.48
CLK4 Q9HAZ1 2/20 0.48
STK17A Q9UEE5 2/20 0.48
MAP4K5 Q9Y4K4 2/20 0.48
DYRK3 O43781 1/20 0.48
RPS6KB1 P23443 1/20 0.48
CSNK2A1 P68400 1/20 0.48
PKN2 Q16513 1/20 0.48
BRSK1 Q8TDC3 1/20 0.48
HIPK2 Q9H2X6 1/20 0.48
MKNK2 Q9HBH9 1/20 0.48
CHEK1 O14757 1/20 0.48
LCK P06239 1/20 0.48
CSF1R P07333 1/20 0.48
PHKG2 P15735 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580810 0.90 CHEK1 (0.59) ADORA2AADORA1MAP4K4PIM1PIM3
SCHEMBL3577456 0.89 MAP4K4 (0.59) ADORA2AADORA1MAP4K4PIM1PIM3
SCHEMBL3585981 0.87 ADORA2A (0.55) ADORA2AADORA1MAP4K4PIM1PIM3
SCHEMBL3589367 0.85 MAP4K4 (0.65) ADORA2AADORA1MAP4K4PIM1PIM3
SCHEMBL3578582 0.84 CHEK2 (0.56) ADORA2AADORA1MAP4K4PIM1PIM3
SCHEMBL6948237 0.79 TSHR (0.50) PKN2KDM4EALDH1A1GAA
SCHEMBL3575241 0.79 MAP4K4 (0.72) ADORA2AADORA1MAP4K4PIM1PIM3
SCHEMBL3577822 0.79 MAP4K4 (0.72) ADORA2AADORA1MAP4K4PIM1PIM3
SCHEMBL3580322 0.77 CHEK1 (0.61) ADORA2AADORA1MAP4K4PIM1PIM3
SCHEMBL3574926 0.75 MAPT (0.55) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed