SCHEMBL3591241

SCHEMBL3591241

CN(CCNC(=O)Cn1nc(Cl)c2cccnc21)C1CCCCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.41
NTRK1 P04629 1/20 0.41
FYN P06241 1/20 0.41
RET P07949 1/20 0.41
MET P08581 1/20 0.41
PDGFRB P09619 1/20 0.41
PIM1 P11309 1/20 0.41
FGFR1 P11362 1/20 0.41
PDGFRA P16234 1/20 0.41
LTK P29376 1/20 0.41
MAP2K2 P36507 1/20 0.41
FLT3 P36888 1/20 0.41
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41
CDK8 P49336 1/20 0.41
GSK3B P49841 1/20 0.41
CDK7 P50613 1/20 0.41
CDK9 P50750 1/20 0.41
NEK2 P51955 1/20 0.41
JAK3 P52333 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3591608 0.85 BCHE (0.43) BCHEACHEKMT2AMEN1TP53
SCHEMBL3591234 0.82 P2RX7 (0.45) KMT2AMEN1MAPTCHRNA7TSHR
SCHEMBL3607948 0.78 KMT2A (0.39) BCHEACHEKMT2AMEN1TP53
SCHEMBL3597267 0.78 BCHE (0.41) BCHEACHEKMT2AMEN1TP53
SCHEMBL3591258 0.77 MAPK1 (0.45) BCHEACHEKMT2AMEN1TP53
SCHEMBL3605621 0.74 TRPA1 (0.43) BCHEACHEKMT2AMEN1TP53
SCHEMBL3599800 0.73 HPGD (0.47) BCHEACHEKMT2AMEN1TP53
SCHEMBL3600246 0.71 GAA (0.55) BCHEACHEKMT2AMEN1GAA
SCHEMBL3602593 0.71 TSHR (0.57) BCHEACHEKMT2AMEN1TP53
SCHEMBL3591679 0.70 KMT2A (0.41) CHEK1NTRK1FYNRETMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7807704-B2 Bicyclic, nitrogen-containing compounds modulating CXCR4 and/or CCXCKR2 CHEMOCENTRYX, INC. (US) 2010-10-05 US disclosed
US-20070275965-A1 CXCR4 modulators CHEMOCENTRYX, INC. (US) 2007-11-29 US disclosed
WO-2007115231-A2 CXCR4 MODULATORS CHEMOCENTRYX, INC. (US) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275965-A1 CXCR4 modulators CXCL12, CXCR4, CXCR1 CHEK1 2083/4885NTRK1 1835/4885FYN 2090/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.