SCHEMBL3592428

SCHEMBL3592428

N#Cc1cc(-c2ccc(F)cc2)sc1-c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.41
CYP11B1 P15538 2/20 0.41
CYP11B2 P19099 2/20 0.41
IKBKB O14920 5/20 0.38
CYP1A2 P05177 2/20 0.38
CHUK O15111 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HSD17B1 P14061 1/20 0.38
HSD17B2 P37059 1/20 0.38
ESR1 P03372 2/20 0.37
ESR2 Q92731 2/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30536527 0.82 ESR2 (0.58) HSD17B1HSD17B2ESR1ESR2HDAC6
SCHEMBL6798956 0.79 CDC7 (0.43) PTGS1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL3325856 0.77 IKBKB (0.38) CYP11B1CYP11B2IKBKBCYP1A2CHUK
SCHEMBL30536578 0.76 HSD17B1 (0.50) CYP3A4CYP2C19HSD17B1HSD17B2ESR1
SCHEMBL3597485 0.72 SNCA (0.53) PTGS1IKBKBCYP1A2CHUKCYP3A4
SCHEMBL4075179 0.70 IKBKB (0.51) PTGS1IKBKBCYP1A2CHUKCYP3A4
SCHEMBL30536525 0.69 ESR2 (0.48) CYP3A4CYP2C19HSD17B1HSD17B2ESR1
SCHEMBL30536537 0.69 SNCA (0.44) HSD17B1HSD17B2ESR1ESR2
SCHEMBL3609166 0.69 MAPK14 (0.61) PTGS1MEN1KMT2ANPSR1KDM4E
SCHEMBL3611196 0.69 KDM4E (0.67) IKBKBCYP1A2CHUKCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8835476-B2 Synthesis of novel antimicrobials WU FAN (CA) 2014-09-16 US disclosed
US-20100076028-A1 Design and Synthesis of Novel Antimicrobials WU FAN 2010-03-25 US disclosed
WO-2006092059-A1 DESIGN AND SYNTHESIS OF NOVEL ANTIMICROBIALS WU FAN (CA) 2006-09-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100076028-A1 Design and Synthesis of Novel Antimicrobials MLX, LPXN, TPX2 PTGS1 1164/4885CYP11B1 3020/4885CYP11B2 3654/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.