SCHEMBL3595020

SCHEMBL3595020

CN(CCNC(=O)Cn1ccc2ccccc21)C1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.52
TP53 P04637 2/20 0.52
TSHR P16473 2/20 0.52
LMNA P02545 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MTNR1A P48039 2/20 0.50
MTNR1B P49286 2/20 0.50
CCNE1 P24864 1/20 0.48
CDK2 P24941 1/20 0.48
CDK5 Q00535 1/20 0.48
MAPK1 P28482 3/20 0.44
MAPT P10636 2/20 0.44
IDO1 P14902 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 2/20 0.43
NTSR1 P30989 1/20 0.43
NPY5R Q15761 1/20 0.43
GAA P10253 1/20 0.43
KDM4E B2RXH2 2/20 0.43
CYP3A4 P08684 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3598446 0.87 KDM4E (0.44) HSD17B10TP53TSHRLMNASMN1; SMN2
SCHEMBL3591066 0.85 ALDH1A1 (0.46) HSD17B10TP53TSHRLMNASMN1; SMN2
SCHEMBL3608129 0.85 KDM4E (0.49) HSD17B10TP53TSHRLMNASMN1; SMN2
SCHEMBL3598309 0.84 SMN1; SMN2 (0.43) HSD17B10TP53TSHRSMN1; SMN2MAPT
SCHEMBL3591244 0.84 TSHR (0.42) HSD17B10TP53TSHRLMNASMN1; SMN2
SCHEMBL3601863 0.84 GRIN2B (0.45) HSD17B10TP53TSHRLMNAMAPT
SCHEMBL14397294 0.83 MAPT (0.40) HSD17B10TP53TSHRLMNASMN1; SMN2
SCHEMBL3586421 0.83 TSHR (0.41) HSD17B10TP53TSHRLMNASMN1; SMN2
SCHEMBL3603866 0.83 MEN1 (0.45) HSD17B10TP53TSHRSMN1; SMN2MAPT
SCHEMBL3585618 0.83 MAPT (0.40) HSD17B10TP53TSHRLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7807704-B2 Bicyclic, nitrogen-containing compounds modulating CXCR4 and/or CCXCKR2 CHEMOCENTRYX, INC. (US) 2010-10-05 US disclosed
US-7807704-B2 Bicyclic, nitrogen-containing compounds modulating CXCR4 and/or CCXCKR2 CHEMOCENTRYX, INC. (US) 2010-10-05 US disclosed
US-7807704-B2 Bicyclic, nitrogen-containing compounds modulating CXCR4 and/or CCXCKR2 CHEMOCENTRYX, INC. (US) 2010-10-05 US disclosed
US-20070275965-A1 CXCR4 modulators CHEMOCENTRYX, INC. (US) 2007-11-29 US disclosed
US-20070275965-A1 CXCR4 modulators CHEMOCENTRYX, INC. (US) 2007-11-29 US disclosed
US-20070275965-A1 CXCR4 modulators CHEMOCENTRYX, INC. (US) 2007-11-29 US disclosed
WO-2007115231-A2 CXCR4 MODULATORS CHEMOCENTRYX, INC. (US) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275965-A1 CXCR4 modulators CXCL12, CXCR4, CXCR1 HSD17B10 3413/4885TP53 1777/4885TSHR 1277/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.