SCHEMBL3595072

SCHEMBL3595072

NCc1c(-c2ccc(Cl)cc2Cl)ncn1CCc1ccccn1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.46
CYP3A4 P08684 3/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CRHR1 P34998 1/20 0.42
DPP8 Q6V1X1 4/20 0.40
DPP9 Q86TI2 2/20 0.40
MARS1 P56192 2/20 0.38
HRH1 P35367 1/20 0.38
HIF1A Q16665 1/20 0.37
HSD17B10 Q99714 1/20 0.37
RAB9A P51151 1/20 0.37
THRB P10828 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3102939 0.89 DPP4 (0.47) DPP4CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL3604955 0.85 DPP4 (0.48) DPP4CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL3092513 0.84 DPP4 (0.47) DPP4CYP3A4DPP8
SCHEMBL3595829 0.83 CYP3A4 (0.44) DPP4CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL3096850 0.82 DPP4 (0.44) DPP4CYP3A4DPP8
SCHEMBL3600802 0.82 DPP4 (0.44) DPP4DPP8
SCHEMBL3586864 0.82 DPP4 (0.45) DPP4CYP3A4DPP8
SCHEMBL3604409 0.81 DPP4 (0.45) DPP4CYP3A4DPP8
SCHEMBL3585733 0.81 DPP4 (0.46) DPP4CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL3583003 0.81 DPP4 (0.42) DPP4CYP3A4DPP8DPP9MARS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed