Dioxane

Dioxane

SCHEMBL35969

C1COCCO1.CC#N

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetonitrile SCHEMBL11848905 1.00 TTR (0.50)
Dioxane SCHEMBL2549097 1.00 TTR (0.50)
Oxirane SCHEMBL6008970 0.96
Dioxane SCHEMBL5129205 0.87 TTR (0.38)
Acetonitrile SCHEMBL2815212 0.85
Tetrahydrofuran SCHEMBL20135739 0.85 ALDH1A1 (0.57)
Tetrahydrofuran SCHEMBL1041391 0.85
Tetrahydrofuran SCHEMBL509785 0.85
Tetrahydrofuran SCHEMBL29033463 0.85 ALDH1A1 (0.57)
Acetonitrile SCHEMBL35968 0.82 ALDH1A1 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 197 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117903192-A Preparation method of 3-methoxy isoquinoline compound intermediate 上海相辉医药科技有限公司 2024-04-19 CN claimed
CN-113788777-B Method for preparing 1-substituted-3-carbonyl pyrrole 华中科技大学 2023-04-11 CN claimed
CN-113788777-A Method for preparing 1-substituted-3-carbonyl pyrrole 华中科技大学 2021-12-14 CN claimed
EP-3784676-A1 POLYMORPHIC FORMS OF BICTEGRAVIR AND ITS SODIUM SALT Mylan Laboratories Ltd. (IN) 2021-03-03 EP claimed
US-20140238293-A1 Crimping Apparatus ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2014-08-28 US claimed
US-8739379-B2 Crimping apparatus ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2014-06-03 US claimed
US-20110283501-A1 CRIMPING APPARATUS ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2011-11-24 US claimed
US-8015687-B2 Method of inserting self-expandable stent in a sheath ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2011-09-13 US claimed
US-8011078-B2 Method of producing stent-balloon assembly ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2011-09-06 US claimed
JP-4733109-B2 2011-07-27 JP claimed
US-20100192353-A1 Method of Producing Stent-Balloon Assembly PACETTI STEPHEN DIRK 2010-08-05 US claimed
US-20100115755-A1 Method of Inserting Self-Expandable Stent in a Sheath PACETTI STEPHEN DIRK 2010-05-13 US claimed
JP-2008500967-A 2008-01-17 JP claimed
US-7235676-B2 Catalytic process for the preparation of epoxides from alkenes COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2007-06-26 US claimed
EP-1732910-A1 AN IMPROVED CATALYTIC PROCESS FOR THE PREPARATION OF EPOXIDES FROM ALKENES Council of Scientific and Industrial Research (IN) 2006-12-20 EP claimed
WO-2005095370-A1 AN IMPROVED CATALYTIC PROCESS FOR THE PREPARATION OF EPOXIDES FROM ALKENES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2005-10-13 WO claimed
US-20050222440-A1 Catalytic process for the preparation of epoxides from alkenes COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2005-10-06 US claimed
CN-1093370-A A kind of new azido erythromycin crystal and preparation method thereof JICAI MEDICINE RESEARCH INST B (CN) 1994-10-12 CN claimed
EP-0005524-A1 Omega-(1,3-dithiolan-2-imino)substituted acetic acids, process for their preparation and pharmaceutical compositions containing them MERRELL DOW PHARMACEUTICALS, INC. (US) 1979-11-28 EP claimed
CN-117447481-A Amorphous substance of Martinib-pyroglutamate and preparation method and application thereof 潍坊医学院 2024-01-26 CN disclosed
US-20240018121-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMCIAL DIVERSITY CENTER, INC. (US) 2024-01-18 US disclosed
US-11691967-B2 Antibiotics effective for gram-negative pathogens THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-07-04 US disclosed
CN-113788777-B Method for preparing 1-substituted-3-carbonyl pyrrole 华中科技大学 2023-04-11 CN disclosed
CN-115521223-A Method for recycling unsymmetrical dimethylhydrazine waste liquid 西安航洁化工科技有限责任公司 2022-12-27 CN disclosed
EP-4058455-A1 NOVEL FUNCTIONALIZED LACTAMS AS MODULATORS OF THE 5-HYDROXYTRYPTAMINE RECEPTOR 7 AND THEIR METHOD OF USE Temple University - Of The Commonwealth System of Higher Education (US) 2022-09-21 EP disclosed
EP-4028130-A1 BENZYL AMINE-CONTAINING 5,6-HETEROAROMATIC COMPOUNDS USEFUL AGAINST MYCOBACTERIAL INFECTION Shionogi & Co., Ltd (JP) 2022-07-20 EP disclosed
CN-113788777-A Method for preparing 1-substituted-3-carbonyl pyrrole 华中科技大学 2021-12-14 CN disclosed
US-20210355137-A1 POLYMORPHIC FORMS OF BICTEGRAVIR AND ITS SODIUM SALT MYLAN LABORATORIES LIMITED (IN) 2021-11-18 US disclosed
WO-2021097116-A1 NOVEL FUNCTIONALIZED LACTAMS AS MODULATORS OF THE 5-HYDROXYTRYPTAMINE RECEPTOR 7 AND THEIR METHOD OF USE TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2021-05-20 WO disclosed
CN-109970714-B Tetradentate platinum (II) complex and application thereof 广东阿格蕾雅光电材料有限公司 2021-04-13 CN disclosed
WO-2021050708-A1 BENZYL AMINE-CONTAINING 5,6-HETEROAROMATIC COMPOUNDS USEFUL AGAINST MYCOBACTERIAL INFECTION SHIONOGI & CO., LTD. (JP) 2021-03-18 WO disclosed
EP-3784676-A1 POLYMORPHIC FORMS OF BICTEGRAVIR AND ITS SODIUM SALT Mylan Laboratories Ltd. (IN) 2021-03-03 EP disclosed
CN-109980111-B Organic electroluminescent device containing tetradentate platinum (II) complex 广东阿格蕾雅光电材料有限公司 2021-02-19 CN disclosed
US-20210017165-A1 ANTIBIOTICS EFFECTIVE FOR GRAM-NEGATIVE PATHOGENS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2021-01-21 US disclosed
US-20200369665-A1 IMIDAZO[1,2-A]PYRAZINE MODULATORS OF THE ADENOSINE A2A RECEPTOR Ryvu Therapeutics S.A. (PL) 2020-11-26 US disclosed
CN-111735781-A Triphenylamine grafted ruthenium complex ratio luminescence pH sensor 北京师范大学 2020-10-02 CN disclosed
CN-108088929-B Analysis method of L-phenylglycine ethyl dane potassium salt 天津大学 2020-05-29 CN disclosed
CN-108350307-B The manufacturing method of metal surface treating composition, metal material 日本帕卡濑精株式会社 2019-11-05 CN disclosed
CN-110325518-A Thiazolium compounds and herbicide 日本欧爱特农业科技株式会社 2019-10-11 CN disclosed
US-20190142798-A1 POLYMER-DES-ETHYL SUNITINIB CONJUGATES NEKTAR THERAPEUTICS 2019-05-16 US disclosed
EP-3283481-B1 CHROMENE DERIVATIVES AS PHOSHOINOSITIDE 3-KINASES INHIBITORS CHIESI FARM SPA (IT) 2019-03-13 EP disclosed
US-10220020-B2 Polymer-des-ethyl sunitinib conjugates NEKTAR THERAPEUTICS (US) 2019-03-05 US disclosed
CN-105001114-B Prepare the new method of Iopromide 沈阳中海生物技术开发有限公司 2018-11-20 CN disclosed
CN-105017063-B 5- amino -2,4,6- triiodo isophthalic acid derivatives and its salt, hydrate or solvate 沈阳中海生物技术开发有限公司 2018-11-20 CN disclosed
CN-108350307-A The manufacturing method of metal surface treating composition, metal material 日本帕卡濑精株式会社 2018-07-31 CN disclosed
CN-108088929-A A kind of analysis method of L-Phenylglycine ethyl dane potassium salts 华北制药股份有限公司 2018-05-29 CN disclosed
US-9968604-B2 Chromene derivatives as phoshoinositide 3-kinases inhibitors CHIESI FARMACEUTICI S.P.A. (IT) 2018-05-15 US disclosed
US-9949854-B2 Crimping method ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2018-04-24 US disclosed
CN-104781288-B Process for producing terminal-modified polybutadiene or terminal-modified hydrogenated polybutadiene, and composition containing same 日本曹达株式会社 2018-04-20 CN disclosed
EP-3283481-A1 CHROMENE DERIVATIVES AS PHOSHOINOSITIDE 3-KINASES INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2018-02-21 EP disclosed
CN-107501542-A A kind of preparation method of Amino End Group polyethylene glycol t-butyl carbamate 湖南华腾制药有限公司 2017-12-22 CN disclosed
CN-104093737-B Antibodies specific for trans-resveratrol and uses thereof IP科技有限公司 2017-11-21 CN disclosed
US-20170326148-A1 PREVENTION OR TREATMENT OF URIC ACID OR GOUT DISEASE Shanton Pharma Pte. Ltd. (SG) 2017-11-16 US disclosed
EP-2654797-B1 POLYMER-DES-ETHYL SUNITINIB CONJUGATES NEKTAR THERAPEUTICS (US) 2017-11-08 EP disclosed
WO-2017171239-A1 ION EXCHANGE SEPARATION MEMBRANE, ELECTROCHEMICAL CELL INCLUDING SAME, FLOW CELL AND FUEL CELL, AND MANUFACTURING METHOD THEREOF 주식회사 엘지화학 2017-10-05 WO disclosed
US-20170252191-A1 CRIMPING METHOD ABBOTT CARDIOVASCULAR SYSTEMS INC (US) 2017-09-07 US disclosed
US-20170202839-A1 Crystalline Form of Pemirolast RSPR PHARMA AB (SE) 2017-07-20 US disclosed
US-9675484-B2 Crimping method ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2017-06-13 US disclosed
US-20170146524-A1 ANTIBODY SPECIFIC FOR TRANS-RESVERATROL AND USE THEREOF IP SCIENCE LIMITED (GB) 2017-05-25 US disclosed
EP-3141549-A1 CRYSTALLINE FORM OF PEMIROLAST FOR USE IN THE TREATMENT OF INFLAMMATIONS RSPR Pharma AB (SE) 2017-03-15 EP disclosed
CN-105102415-B Method for improving optical purity of 2-hydroxycarboxylic acid or derivative thereof 兴和株式会社 2017-03-15 CN disclosed
US-9547001-B2 Antibody specific for trans-resveratrol and use thereof IP SCIENCE LIMITED (GB) 2017-01-17 US disclosed
CN-106317099-A Aminoalkylalkoxydisiloxane compound and method for preparing the same 信越化学工业株式会社 2017-01-11 CN disclosed
EP-2443120-B1 CRYSTALLINE FORM OF PEMIROLAST RSPR PHARMA AB (SE) 2016-11-02 EP disclosed
US-20160303123-A1 CHROMENE DERIVATIVES AS PHOSHOINOSITIDE 3-KINASES INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2016-10-20 US disclosed
WO-2016166239-A1 CHROMENE DERIVATIVES AS PHOSHOINOSITIDE 3-KINASES INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2016-10-20 WO disclosed
US-20160278956-A1 CRIMPING METHOD ABBOTT CARDIOVASCULAR SYSTEMS INC (US) 2016-09-29 US disclosed
EP-2776464-B1 ANTIBODY SPECIFIC FOR TRANS-RESVERATROL AND USE THEREOF IP SCIENCE LTD (GB) 2016-09-28 EP disclosed
US-20160250217-A1 CRYSTALLINE FORM OF PEMIROLAST RSPR PHARMA AB (SE) 2016-09-01 US disclosed
US-9388172-B2 Substituted carbamate compounds HOFFMANN-LA ROCHE INC. (US) 2016-07-12 US disclosed
CN-103717593-B Regulate kinase whose compositions and method 克勒韦谢尔制药公司 2016-07-06 CN disclosed
CN-105732635-A Toll-like receptor 7 agonist 南京明德新药研发股份有限公司 2016-07-06 CN disclosed
US-9375334-B2 Crimping method ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2016-06-28 US disclosed
EP-2718290-B1 COMPOSITIONS AND METHODS FOR MODULATING A KINASE CLEVEXEL PHARMA (FR) 2016-05-04 EP disclosed
CN-105017063-A 5-amino-2,4,6-triiodo m-phthalic acid derivative and salt, hydrate or solvate J&HEALTH BIOTECHNOLOGY CO LTD 2015-11-04 CN disclosed
CN-105001114-A New method for preparing iopromide J&HEALTH BIOTECHNOLOGY CO LTD 2015-10-28 CN disclosed
US-20150282969-A1 Crimping Method ABBOTT CARDIOVASCULAR SYSTEMS (US) 2015-10-08 US disclosed
EP-2917208-A1 [3-HETEROARYL-2-TRIFLUOROMETHYL-PROPYL]-PIPERIDIN-1-YLE OR -MORPHOLIN-4-YLE COMPOUNDS AS TRPA1 ANTAGONISTS FOR THE TREATMENT OF RESPIRATORY DISEASES F. Hoffmann-La Roche AG (CH) 2015-09-16 EP disclosed
US-20150239873-A1 SUBSTITUTED CARBAMATE COMPOUNDS HOFFMANN-LA ROCHE INC. (US) 2015-08-27 US disclosed
WO-2015082592-A2 METHOD FOR PREPARING AMINOARYLBORANE COMPOUNDS OR DERIVATIVES THEREOF Universite de Bordeaux (FR) 2015-06-11 WO disclosed
EP-2881398-A1 Method for preparing aminoarylborane compounds or derivatives thereof Université de Bordeaux I (FR) 2015-06-10 EP disclosed
US-9044312-B2 Crimping method ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2015-06-02 US disclosed
US-9006431-B2 Crystalline form of pemirolast RSPR PHARMA AB (SE) 2015-04-14 US disclosed
US-8937065-B2 Compositions and methods for modulating a kinase CLEVEXEL PHARMA (FR) 2015-01-20 US disclosed
US-20140349319-A1 ANTIBODY SPECIFIC FOR TRANS-RESVERATROL AND USE THEREOF IP SCIENCE LIMITED (GB) 2014-11-27 US disclosed
US-20140329839-A1 New Crystalline Form of Pemirolast CARDOZ AB (SE) 2014-11-06 US disclosed
CN-104093737-A Antibodies specific for trans-resveratrol and uses thereof IP SCIENCE LTD 2014-10-08 CN disclosed
EP-2776464-A1 ANTIBODY SPECIFIC FOR TRANS - RESVERATROL AND USE THEREOF IP Science Limited (GB) 2014-09-17 EP disclosed
US-20140238293-A1 Crimping Apparatus ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2014-08-28 US disclosed
EP-2768810-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2014-08-27 EP disclosed
US-8739379-B2 Crimping apparatus ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2014-06-03 US disclosed
EP-2079845-B1 Process for producing vessels containing bacterial cellulose ARTERION AB (SE) 2014-05-21 EP disclosed
WO-2014072325-A1 [3-HETEROARYL-2-TRIFLUOROMETHYL-PROPYL]-PIPERIDIN-1-YLE OR -MORPHOLIN-4-YLE COMPOUNDS AS TRPA1 ANTAGONISTS FOR THE TREATMENT OF RESPIRATORY DISEASES F. HOFFMANN-LA ROCHE AG (CH) 2014-05-15 WO disclosed
EP-2718290-A2 COMPOSITIONS AND METHODS FOR MODULATING A KINASE Clevexel Pharma (FR) 2014-04-16 EP disclosed
US-20140039030-A1 POLYMER-DES-ETHYL SUNITINIB CONJUGATES NEKTAR THERAPEUTICS (US) 2014-02-06 US disclosed
EP-2654797-A1 POLYMER-DES-ETHYL SUNITINIB CONJUGATES Nektar Therapeutics (US) 2013-10-30 EP disclosed
WO-2013136296-A2 WATER-SOLUBLE ORGANOMETALLIC RUTHENIUM AND IRON COMPUNDS PRESENTING HETEROAROMATIC LIGANDS UNIVERSIDADE DE LISBOA (PT) 2013-09-19 WO disclosed
WO-2013068758-A1 ANTIBODY SPECIFIC FOR TRANS - RESVERATROL AND USE THEREOF IP SCIENCE LIMITED (GB) 2013-05-16 WO disclosed
WO-2013059666-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA, INC. (US) 2013-04-25 WO disclosed
WO-2012172438-A9 COMPOSITIONS AND METHODS FOR MODULATING A KINASE DYNAMIX PHARMACEUTICALS LTD. (IL) 2013-02-07 WO disclosed
WO-2012172438-A2 COMPOSITIONS AND METHODS FOR MODULATING A KINASE DYNAMIX PHARMACEUTICALS LTD. (IL) 2012-12-20 WO disclosed
US-20120316148-A1 Compositions and Methods for Modulating a Kinase DYNAMIX PHARMACEUTICALS LTD. (IL) 2012-12-13 US disclosed
US-8273706-B2 Isobarically labeled analytes and fragment ions derived therefrom DH TECHNOLOGIES DEVELOPMENT PTE. LTD. (SG) 2012-09-25 US disclosed
US-20120220558-A1 Methods of Treating Hormone-Related Conditions Using Thio-Oxindole Derivatives WYETH LLC (US) 2012-08-30 US disclosed
US-8242098-B2 Methods of treating hormone-related conditions using thio-oxindole derivatives WYETH LLC (US) 2012-08-14 US disclosed
WO-2012088522-A1 POLYMER-DES-ETHYL SUNITINIB CONJUGATES NEKTAR THERAPEUTICS (US) 2012-06-28 WO disclosed
US-20120157415-A1 New Crystalline Form of Pemirolast CARDOZ AB (SE) 2012-06-21 US disclosed
WO-2010146348-A9 CRYSTALLINE FORM OF PEMIROLAST CARDOZ AB (SE) 2012-05-03 WO disclosed
EP-2443120-A2 NEW CRYSTALLINE FORM OF PEMIROLAST Cardoz AB (SE) 2012-04-25 EP disclosed
EP-2426211-A1 Bacterial cellulose tubes Arterion AB (SE) 2012-03-07 EP disclosed
US-20110283501-A1 CRIMPING APPARATUS ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2011-11-24 US disclosed
US-8020273-B2 High humidity crimping process ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2011-09-20 US disclosed
US-8015684-B2 Crimping apparatus ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2011-09-13 US disclosed
US-8015687-B2 Method of inserting self-expandable stent in a sheath ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2011-09-13 US disclosed
US-8011078-B2 Method of producing stent-balloon assembly ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2011-09-06 US disclosed
EP-1405922-B1 Substrates for beta-lactamase and uses thereof UNIV CALIFORNIA (US) 2011-08-24 EP disclosed
WO-2010146348-A2 NEW CRYSTALLINE FORM OF PEMIROLAST CARDOZ AB (SE) 2010-12-23 WO disclosed
WO-2010146341-A2 NEW CRYSTALLINE FORM OF PEMIROLAST CARDOZ AB (SE) 2010-12-23 WO disclosed
EP-2251334-A1 Labeling reagents and labeled analytes Life Technologies Corporation (US) 2010-11-17 EP disclosed
EP-2229397-A2 PROCESS FOR PREPARING RISEDRONATE SODIUM AS ANHYDROUS AND HYDRATE FORMS Dongwoo Syntech Co., Ltd. (KR) 2010-09-22 EP disclosed
EP-1701945-B1 LABELING REAGENTS, LABELED ANALYTES, INCLUDING MIXTURES THEREOF, AND FRAGMENT IONS DERIVED THEREFROM AND METHODS FOR THE ANALYSIS THEREOF LIFE TECHNOLOGIES CORP (US) 2010-09-01 EP disclosed
US-20100192353-A1 Method of Producing Stent-Balloon Assembly PACETTI STEPHEN DIRK 2010-08-05 US disclosed
US-20100129842-A1 ISOBARICALLY LABELED ANALYTES AND FRAGMENT IONS DERIVED THEREFROM Life Technologies Corporation (US) 2010-05-27 US disclosed
US-20100122446-A1 Crimping Apparatus PACETTI STEPHEN DIRK 2010-05-20 US disclosed
US-20100115759-A1 High Humidity Crimping Process PACETTI STEPHEN DIRK 2010-05-13 US disclosed
US-20100115755-A1 Method of Inserting Self-Expandable Stent in a Sheath PACETTI STEPHEN DIRK 2010-05-13 US disclosed
US-7673379-B1 providing a stent having a polymeric component, wherein the polymeric component is a phosphoryl choline acrylate polymer, exposing the stent to a relative humidity of 20% to 100%, and crimping the stent on a balloon of a catheter assembly ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2010-03-09 US disclosed
US-20100042197-A1 PREPARATION OF HOLLOW CELLULOSE VESSELS ARTERION AB (SE) 2010-02-18 US disclosed
EP-2079845-A2 ARTIFICIAL VESSELS Arterion AB (SE) 2009-07-22 EP disclosed
WO-2009072769-A2 PROCESS FOR PREPARING RISEDRONATE SODIUM AS ANHYDROUS AND HYDRATE FORMS DONGWOO SYNTECH CO., LTD (KR) 2009-06-11 WO disclosed
US-20090099223-A1 METHODS OF TREATING HORMONE-RELATED CONDITIONS USING THIO-OXINDOLE DERIVATIVES WYETH (US) 2009-04-16 US disclosed
US-7488734-B2 Methods of treating hormone-related conditions using thio-oxindole derivatives WYETH (US) 2009-02-10 US disclosed
EP-1077686-B1 EXTERNALLY TRIGGERED MICROCAPSULES NASA JOHNSON SPACE CT (US) 2008-08-06 EP disclosed
WO-2008040729-A2 PROCESS FOR THE PREPARATION OF HOLLOW CELLULOSE VESSELS BY CULTURING CELLULOSE- PRODUCING MICROORGANISMS ON THE SURFACE OF A HOLLOW CARRIER AND PROVIDING A GAS HAVING AN OXYGEN LEVEL OF AT LEAST 35% ARTERION AB (SE) 2008-04-10 WO disclosed
US-7235676-B2 Catalytic process for the preparation of epoxides from alkenes COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2007-06-26 US disclosed
EP-1732910-A1 AN IMPROVED CATALYTIC PROCESS FOR THE PREPARATION OF EPOXIDES FROM ALKENES Council of Scientific and Industrial Research (IN) 2006-12-20 EP disclosed
US-7115649-B2 Methods of treating skin disorders using thio-oxindole derivatives WYETH (US) 2006-10-03 US disclosed
EP-1701945-A1 LABELING REAGENTS, LABELED ANALYTES, INCLUDING MIXTURES THEREOF, AND FRAGMENT IONS DERIVED THEREFROM AND METHODS FOR THE ANALYSIS THEREOF Applera Corporation (US) 2006-09-20 EP disclosed
US-7091234-B2 Thio-oxindole derivatives WYETH (US) 2006-08-15 US disclosed
WO-2005095370-A1 AN IMPROVED CATALYTIC PROCESS FOR THE PREPARATION OF EPOXIDES FROM ALKENES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2005-10-13 WO disclosed
US-20050222440-A1 Catalytic process for the preparation of epoxides from alkenes COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2005-10-06 US disclosed
EP-1531806-A4 USE OF THIO-OXINDOLE DERIVATIVES IN TREATMENT OF HORMONE-RELATED CONDITIONS WYETH CORP (US) 2005-09-21 EP disclosed
EP-1515680-A4 USE OF THIO-OXINDOLE DERIVATIVES IN TREATMENT OF SKIN DISORDERS WYETH CORP (US) 2005-09-21 EP disclosed
US-6946454-B2 Thio-oxindole derivatives WYETH (US) 2005-09-20 US disclosed
CN-1662206-A Use of thio-2-oxindole derivatives in treatment of skin disorders WYETH CORP (US) 2005-08-31 CN disclosed
US-20050171186-A1 3-(1',2'-Dihydro-2'-thioxospiro[cyclohexane-1,3'-[3H]indol]-5'-yl)benzonitrile; 5'-(5-Cyano-1-methyl-1H-pyrrol-2-yl)spiro[cyclohexane-1,3'-[3H]indol]-2'-ylidenecyanamide; progesterone receptor agonist; mixture with estrone (estrogen); hormone replacement therapy, contraception; anticarcinogenic WYETH (US) 2005-08-04 US disclosed
WO-2005068446-A1 LABELING REAGENTS, LABELED ANALYTES, INCLUDING MIXTURES THEREOF, AND FRAGMENT IONS DERIVED THEREFROM AND METHODS FOR THE ANALYSIS THEREOF APPLERA CORPORATION (US) 2005-07-28 WO disclosed
US-20050148087-A1 Isobarically labeled analytes and fragment ions derived therefrom APPLERA CORPORATION 2005-07-07 US disclosed
US-20050147985-A1 Mixtures of isobarically labeled analytes and fragments ions derived therefrom APPLERA CORPORATION 2005-07-07 US disclosed
EP-1531806-A2 USE OF THIO-OXINDOLE DERIVATIVES IN TREATMENT OF HORMONE-RELATED CONDITIONS Wyeth (US) 2005-05-25 EP disclosed
US-6875765-B2 Arylsulfonamide ethers, and methods of use thereof WARNER-LAMBERT COMPANY (US) 2005-04-05 US disclosed
EP-1515680-A2 USE OF THIO-OXINDOLE DERIVATIVES IN TREATMENT OF SKIN DISORDERS Wyeth (US) 2005-03-23 EP disclosed
US-20050054711-A1 Thio-oxindole derivatives WYETH 2005-03-10 US disclosed
US-6841568-B2 Thio-oxindole derivatives WYETH (US) 2005-01-11 US disclosed
US-20040006122-A1 Methods of treating skin disorders using thio-oxindole derivatives WYETH 2004-01-08 US disclosed
US-20040002535-A1 Methods of treating hormone-related conditions using thio-oxindole derivatives WYETH (US) 2004-01-01 US disclosed
WO-2004000225-A2 USE OF THIO-OXINDOLE DERIVATIVES IN TREATMENT OF HORMONE-RELATED CONDITIONS WYETH (US) 2003-12-31 WO disclosed
WO-2004000227-A2 USE OF THIO-OXINDOLE DERIVATIVES IN TREATMENT OF SKIN DISORDERS WYETH (US) 2003-12-31 WO disclosed
US-20030225109-A1 Thio-oxindole derivatives WYETH (US) 2003-12-04 US disclosed
US-6583145-B1 Thio-oxindole derivatives WYETH 2003-06-24 US disclosed
US-20030096826-A1 Arylsulfonamide ethers, and methods of use thereof WARNER-LAMBERT COMPANY 2003-05-22 US disclosed
US-20030064978-A1 Novel compounds ASTRAZENECA AB. (SE) 2003-04-03 US disclosed
US-6521657-B2 Indole derivatives which are agonists of the progesterone receptor and useful for treatment of carcinoma and adenocarcinomas of uterine leiomyomata, endometriosis or polycystic ovary syndorme in a mammal WYETH 2003-02-18 US disclosed
US-20020169198-A1 Thio-oxindole derivatives WYETH (US) 2002-11-14 US disclosed
US-20020103248-A1 Thio-oxindole derivatives WYETH LLC 2002-08-01 US disclosed
WO-2002028808-A1 TRIPTYCENE ANALOGS KANSAS STATE UNIVERSITY RESEARCH FOUNDATION (US) 2002-04-11 WO disclosed
US-6355648-B1 COMPOUNDS AS CONTRACEPTIVES AND PROGESTERONE ANTAGONIST AMERICAN HOME PRODUCTS CORPORATION 2002-03-12 US disclosed
EP-1181275-A1 THIO-OXINDOLE DERIVATIVES American Home Products Corporation (US) 2002-02-27 EP disclosed
US-6297231-B1 CARBOXYLATION OF NITROGEN IN PYRROLIDINE RING TO RENDER RESISTANT TO BETA-LACTAMASES MERCK & CO., INC. 2001-10-02 US disclosed
US-6248916-B1 WATER SOLUBLE, STRAIGHT CHAIN BORON-RICH OLIGOPHOSPHATE WHICH COMPRISES AN ORDERED PLURALITY OF CARBORANE MONOMER UNITS HAVING TWO HYDROXYL GROUPS ATTACHED THERETO BEING LINKED BY THE HYDROXYL GROUPS TO PHOSPHATE UNITS REGENTS OF THE UNIVERSITY OF CALIFORNIA 2001-06-19 US disclosed
EP-0937079-A4 STABILIZED CARBAPENEM ANTIBIOTIC COMPOSITIONS AND METHOD OF MAKING MERCK & CO INC (US) 2001-01-24 EP disclosed
WO-2000066555-A1 THIO-OXINDOLE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-11-09 WO disclosed
WO-2000008026-A2 FUNGICIDAL FUSED BICYCLIC HETEROCYCLES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2000-02-17 WO disclosed
EP-0937079-A1 STABILIZED CARBAPENEM ANTIBIOTIC COMPOSITIONS AND METHOD OF MAKING Merck &amp; Co., Inc. (a New Jersey corp.) (US) 1999-08-25 EP disclosed
US-5856551-A REACTING DIHYDROXYCARBORANE WITH PHOSPHORUS COUPLING AGENT;THEN ALCOHOL THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1999-01-05 US disclosed
WO-1998018800-A1 STABILIZED CARBAPENEM ANTIBIOTIC COMPOSITIONS AND METHOD OF MAKING MERCK & CO., INC. (US) 1998-05-07 WO disclosed
EP-0514917-B1 Process for and 2-(cyanoimino)-quinazoline derivatives useful as intermediates in the preparation of 6,7-di-(chloro)-1,5-di(hydro)-imidazo-[2,1-b]quinazolin-2[3H]-one and process for preparing the 2-(cyanoimino)-quinazoline derivatives EGYT GYOGYSZERVEGYESZETI GYAR (HU) 1996-12-27 EP disclosed
WO-1995026359-A1 MACROMOLECULAR STRUCTURES FOR BORON NEUTRON-CAPTURE THERAPY REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-10-05 WO disclosed
US-5426244-A Para-selective; reacting a phenol with hydrogen peroxide in presence of crystalline titanosilicate catalyst and cyclic ether MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1995-06-20 US disclosed
US-5391737-A Process for the preparation of 6,7-dichloro-1,5-dihydroimidazo[2,1-b]quinazolin-2[3H]-one EGIS GYOGYSZERGYAR (HU) 1995-02-21 US disclosed
EP-0420248-B1 Absorbent structures KIMBERLY CLARK CO (US) 1994-03-09 EP disclosed
EP-0514917-A1 Process for and 2-(cyanoimino)-quinazoline derivatives useful as intermediates in the preparation of 6,7-di-(chloro)-1,5-di(hydro)-imidazo-[2,1-b]quinazolin-2[3H]-one and process for preparing the 2-(cyanoimino)-quinazoline derivatives EGIS GYOGYSZERGYAR (HU) 1992-11-25 EP disclosed
EP-0258662-B1 COLOR PHOTOGRAPHS AND METHOD FOR PREPARATION OF THE SAME FUJI PHOTO FILM CO., LTD. (JP) 1992-05-27 EP disclosed
US-5082723-A Diapers, sanitayr napkins KIMBERLY-CLARK CORPORATION (US) 1992-01-21 US disclosed
EP-0420248-A1 Absorbent structures KIMBERLY-CLARK CORPORATION (US) 1991-04-03 EP disclosed
US-4976891-A Antithrombotic, antivasoconstricting, antibronchoconstricting SHIONOGI & CO., LTD. (JP) 1990-12-11 US disclosed
US-4960909-A ANTICOAGULANTS; VASODILATORS; BRONCHODILATOR AGENTS SHIONOGI & CO., LTD. (JP) 1990-10-02 US disclosed
EP-0221996-B1 SUBSTITUTED 2,3-DIHYDRO-6-HYDROXY-PYRIMIDO [2,1-f] PURINE-4,8(1H,9H)-DIONES SCHERING CORPORATION (US) 1990-08-29 EP disclosed
CN-1008737-B Process for preparing benzo [1] oxy [5] thiacycloheptene derivatives TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1990-07-11 CN disclosed
US-4920152-A Crosslinking adsorbed coating with hydrophobic reagent PURDUE RESEARCH FOUNDATION (US) 1990-04-24 US disclosed
EP-0335390-A2 Novel cephalosporin compounds SAGAMI CHEMICAL RESEARCH CENTER (JP) 1989-10-04 EP disclosed
EP-0258662-A2 Color photographs and method for preparation of the same FUJI PHOTO FILM CO., LTD. (JP) 1988-03-09 EP disclosed
EP-0221996-A1 SUBSTITUTED 2,3-DIHYDRO-6-HYDROXY-PYRIMIDO [2,1-f] PURINE-4,8(1H,9H)-DIONES. SCHERING CORP (US) 1987-05-20 EP disclosed
WO-1986006724-A1 SUBSTITUTED 2,3-DIHYDRO-6-HYDROXY-PYRIMIDO AD2,1-f BD-PURINE-4,8(1H,9H)-DIONES SCHERING CORPORATION (US) 1986-11-20 WO disclosed
US-4435533-A FIREPROOFING; WRINKLE RESISTANCE TSOLIS ALEXANDROS K 1984-03-06 US disclosed
US-4216206-A Antibiotics S 53210/A-I, S 53210/A-II and S 53210/A-III SANDOZ LTD. (CH) 1980-08-05 US disclosed
EP-0008442-A2 2-Lower alkyl-7-substituted-2 or 3-cephem-4-carboxylic acid compounds, processes for their preparation and pharmaceutical compositions containing them FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1980-03-05 EP disclosed
EP-0008442-A2 2-Lower alkyl-7-substituted-2 or 3-cephem-4-carboxylic acid compounds, processes for their preparation and pharmaceutical compositions containing them FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1980-03-05 EP disclosed