SCHEMBL3597097

SCHEMBL3597097

CC(O)Cn1cnc(-c2ccc(Cl)cc2Cl)c1CN

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 12/20 0.45
DPP8 Q6V1X1 4/20 0.45
CYP3A4 P08684 2/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HIF1A Q16665 1/20 0.36
CRHR1 P34998 2/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3596963 0.83 DPP4 (0.58) DPP4DPP8CYP3A4
SCHEMBL3603728 0.83 DPP4 (0.45) DPP4DPP8CYP3A4TP53CYP1A2
SCHEMBL3096567 0.82 DPP4 (0.46) DPP4DPP8CYP3A4
SCHEMBL3598301 0.82 DPP4 (0.48) DPP4DPP8CYP3A4CYP2C19
SCHEMBL3600930 0.81 DPP4 (0.46) DPP4DPP8CYP3A4CRHR1
SCHEMBL3091767 0.81 DPP4 (0.50) DPP4DPP8CRHR1
SCHEMBL4660649 0.81 DPP4 (0.48) DPP4DPP8CYP3A4
SCHEMBL3600399 0.80 DPP4 (0.42) DPP4DPP8CYP3A4CRHR1
SCHEMBL3091375 0.80 DPP4 (0.47) DPP4DPP8CYP3A4TP53
SCHEMBL3603864 0.79 DPP4 (0.42) DPP4DPP8CYP3A4TP53CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed