SCHEMBL3598301

SCHEMBL3598301

NCc1c(-c2ccc(Cl)cc2Cl)ncn1CC(c1ccccc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 14/20 0.48
CYP3A4 P08684 3/20 0.42
DPP8 Q6V1X1 5/20 0.41
OPRM1 P35372 1/20 0.39
OPRK1 P41145 1/20 0.39
DPP9 Q86TI2 2/20 0.37
CNR1 P21554 1/20 0.37
HSP90AB1 P08238 1/20 0.37
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3598381 0.88 DPP4 (0.49) DPP4CYP3A4DPP8OPRM1OPRK1
SCHEMBL3079559 0.84 DPP4 (0.51) DPP4CYP3A4DPP8DPP9CNR1
SCHEMBL3597097 0.82 DPP4 (0.45) DPP4CYP3A4DPP8CYP2C19
SCHEMBL3604955 0.81 DPP4 (0.48) DPP4CYP3A4DPP8DPP9CNR1
SCHEMBL3595249 0.80 DPP4 (0.47) DPP4CYP3A4DPP8DPP9CYP2C19
SCHEMBL3596963 0.80 DPP4 (0.58) DPP4CYP3A4DPP8DPP9
SCHEMBL4660649 0.80 DPP4 (0.48) DPP4CYP3A4DPP8
SCHEMBL3084580 0.80 DPP4 (0.49) DPP4CYP3A4DPP8CNR1
SCHEMBL3585733 0.79 DPP4 (0.46) DPP4CYP3A4DPP8DPP9CNR1
SCHEMBL3601689 0.79 DPP4 (0.46) DPP4CYP3A4DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed