SCHEMBL3598377

SCHEMBL3598377

NCc1c(-c2ccc(Cl)cc2Cl)ncn1CCN1CCCC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 8/20 0.43
HTT P42858 1/20 0.42
ATM Q13315 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
DPP8 Q6V1X1 5/20 0.41
CNR1 P21554 2/20 0.40
CNR2 P34972 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
MCHR1 Q99705 1/20 0.39
SIGMAR1 Q99720 2/20 0.39
CRHR1 P34998 2/20 0.38
KCNH2 Q12809 1/20 0.37
TGFBR1 P36897 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3598863 0.99 HTT (0.43) DPP4HTTATMTDP1DPP8
SCHEMBL3601192 0.91 TSHR (0.44) DPP4HTTDPP8SIGMAR1TGFBR1
SCHEMBL3600930 0.83 DPP4 (0.46) DPP4DPP8CYP3A4CRHR1
SCHEMBL3091767 0.83 DPP4 (0.50) DPP4DPP8CNR1CRHR1
SCHEMBL3600855 0.81 DPP4 (0.45) DPP4DPP8CYP3A4
SCHEMBL3096850 0.81 DPP4 (0.44) DPP4DPP8CYP3A4
SCHEMBL3596892 0.81 DPP4 (0.44) DPP4DPP8CYP3A4TGFBR1
SCHEMBL3600802 0.81 DPP4 (0.44) DPP4DPP8CNR1
SCHEMBL3596963 0.80 DPP4 (0.58) DPP4DPP8CYP3A4
SCHEMBL4660649 0.80 DPP4 (0.48) DPP4DPP8CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed