SCHEMBL3598381

SCHEMBL3598381

NCc1c(-c2ccc(Cl)cc2Cl)ncn1CCC(c1ccccc1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 11/20 0.49
CYP3A4 P08684 2/20 0.41
DPP8 Q6V1X1 4/20 0.40
MDM4 O15151 1/20 0.38
TP53 P04637 1/20 0.38
MDM2 Q00987 1/20 0.38
HSD11B1 P28845 1/20 0.36
DPP9 Q86TI2 1/20 0.36
CCR5 P51681 1/20 0.36
CNR1 P21554 1/20 0.35
HSP90AB1 P08238 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRK1 P41145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3598301 0.88 DPP4 (0.48) DPP4CYP3A4DPP8DPP9CNR1
SCHEMBL3603728 0.85 DPP4 (0.45) DPP4CYP3A4DPP8MDM4TP53
SCHEMBL3604955 0.84 DPP4 (0.48) DPP4CYP3A4DPP8DPP9CNR1
SCHEMBL3600919 0.83 MDM4 (0.42) DPP4CYP3A4DPP8MDM4TP53
SCHEMBL3079559 0.82 DPP4 (0.51) DPP4CYP3A4DPP8MDM4TP53
SCHEMBL3585733 0.82 DPP4 (0.46) DPP4CYP3A4DPP8DPP9CNR1
SCHEMBL3601689 0.82 DPP4 (0.46) DPP4CYP3A4DPP8
SCHEMBL3603961 0.81 DPP4 (0.46) DPP4CYP3A4DPP8DPP9CNR1
SCHEMBL3590139 0.81 DPP4 (0.46) DPP4CYP3A4DPP8DPP9CNR1
SCHEMBL3091767 0.81 DPP4 (0.50) DPP4DPP8HSD11B1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed