SCHEMBL35988

SCHEMBL35988

c1ccc(CCCc2ccc(-c3cccnc3)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.61
MKNK1 Q9BUB5 2/20 0.61
MKNK2 Q9HBH9 2/20 0.61
CYP3A4 P08684 2/20 0.54
ALDH1A1 P00352 1/20 0.54
CYP1A2 P05177 1/20 0.54
KDR P35968 1/20 0.51
TEK Q02763 1/20 0.51
PTAFR P25105 1/20 0.51
CYP11B1 P15538 2/20 0.50
CYP11B2 P19099 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
GBA1 P04062 2/20 0.49
LMNA P02545 1/20 0.49
ELOVL1 Q9BW60 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP19A1 P11511 1/20 0.49
CYP2C9 P11712 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12435674 0.84 CYP3A4 (0.64) CYP2A6MKNK1MKNK2CYP3A4ALDH1A1
SCHEMBL4966893 0.84 CYP2A6 (0.69) CYP2A6MKNK1MKNK2CYP3A4ALDH1A1
SCHEMBL15060898 0.83 TDP1 (0.67) CYP2A6MKNK1MKNK2CYP3A4ALDH1A1
SCHEMBL14080858 0.83 CYP2A6 (0.67) CYP2A6MKNK1MKNK2CYP3A4ALDH1A1
SCHEMBL8200325 0.83 CYP2A6 (0.68) CYP2A6CYP1A2L3MBTL1CYP2D6
SCHEMBL3400752 0.82 CYP2A6 (0.79) CYP2A6MKNK1MKNK2CYP3A4ALDH1A1
SCHEMBL29468039 0.82 CYP2A6 (0.79) CYP2A6MKNK1MKNK2CYP3A4ALDH1A1
SCHEMBL9826765 0.82 HTR2A (0.62)
SCHEMBL20888564 0.81 CYP2A6 (0.56) CYP2A6MKNK1MKNK2CYP3A4ALDH1A1
SCHEMBL13527201 0.81 TDP1 (0.65) CYP2A6MKNK1MKNK2CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110281822-A1 AROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHONATE (S1P) RECEPTOR ACTIVITY ALLERGAN, INC. (US) 2011-11-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110281822-A1 AROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHONATE (S1P) RECEPTOR ACTIVITY S1PR1, S1PR3, S1PR2 CYP2A6 3025/4885MKNK1 1006/4885MKNK2 1150/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.