SCHEMBL3601893

SCHEMBL3601893

C[C@@H](CC1CCCCC1)N(CN)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 1/20 0.40
CTSK P43235 6/20 0.38
CTSL P07711 3/20 0.38
CTSB P07858 3/20 0.38
CTSH P09668 2/20 0.37
LTA4H P09960 1/20 0.37
CYP2D6 P10635 1/20 0.37
ATM Q13315 1/20 0.36
CPB2 Q96IY4 3/20 0.36
ALOX5 P09917 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15049847 0.82 PSEN1 (0.30)
SCHEMBL23005007 0.74 NPY5R (0.45) NPY5RCTSKCTSLCTSBCYP2D6
SCHEMBL3601888 0.70 NPY5R (0.38) NPY5RCTSKCTSLCTSBCTSH
SCHEMBL19385536 0.70 NPY5R (0.38) NPY5RCTSKCTSLCTSBCTSH
SCHEMBL27182810 0.69 NPY5R (0.43) NPY5RCTSKCTSLCTSBCTSH
SCHEMBL28948946 0.69 LTA4H (0.46) CTSKCTSLCTSBLTA4H
SCHEMBL7794348 0.69 LTA4H (0.46) CTSKCTSLCTSBLTA4H
SCHEMBL5326239 0.69 LTA4H (0.46) CTSKCTSLCTSBLTA4H
SCHEMBL19817250 0.69 LTA4H (0.46) CTSKCTSLCTSBLTA4H
SCHEMBL14947101 0.69 LTA4H (0.46) CTSKCTSLCTSBLTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8455521-B2 Diaminoalkane aspartic protease inhibitors VITAE PHARMACEUTICALS, INC. (US) 2013-06-04 US disclosed
US-7754737-B2 Diaminoalkane aspartic protease inhibitors VITAE PHARMACEUTICALS, INC. (US) 2010-07-13 US disclosed
US-20090018103-A1 Diaminoalkane Aspartic Protease Inhibitors VITAE PHARMACEUTICAL, INC (US) 2009-01-15 US disclosed
EP-1807078-A1 DIAMINOALKANE ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2007-07-18 EP disclosed
WO-2006042150-A1 DIAMINOALKANE ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2006-04-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090018103-A1 Diaminoalkane Aspartic Protease Inhibitors DNPEP, PEPD, ACE NPY5R 2594/4885CTSK 31/4885CTSL 82/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.