SCHEMBL3602567

SCHEMBL3602567

N#Cc1cccc(OC2CCN(C(=O)O)CC2)n1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.55
GPR119 Q8TDV5 2/20 0.43
MDM2 Q00987 1/20 0.41
JAK3 P52333 1/20 0.41
EPHX2 P34913 2/20 0.39
BTK Q06187 2/20 0.39
FFAR4 Q5NUL3 2/20 0.37
SRD5A1 P18405 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
KCNH2 Q12809 1/20 0.36
HRH3 Q9Y5N1 2/20 0.36
SCD O00767 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3601742 0.83 GPR119 (0.63) MGLLGPR119
SCHEMBL3613521 0.81 HRH3 (0.55) MGLLKCNH2HRH3
SCHEMBL5266382 0.81 HRH3 (0.46) GPR119MDM2EPHX2BTKFFAR4
SCHEMBL5267084 0.80 EPHX2 (0.41) MDM2EPHX2BTKFFAR4KCNH2
SCHEMBL5270350 0.80 HCRTR1 (0.44) GPR119MDM2EPHX2BTKKCNH2
SCHEMBL16008245 0.79 GPR119 (0.56) MGLLGPR119
SCHEMBL16008246 0.79 GPR119 (0.56) MGLLGPR119
SCHEMBL25087455 0.79 CTSK (0.45) MGLLFFAR4KCNH2HRH3
SCHEMBL4442024 0.79 HRH3 (0.49) MGLLGPR119MDM2ALDH1A1HRH3
SCHEMBL3602573 0.78 HRH3 (0.43) GPR119EPHX2BTKFFAR4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7723331-B2 Thienopyrimidine compounds and uses thereof ASTRAZENECA AB (SE) 2010-05-25 US disclosed
EP-2121703-A1 THIENOPYRIMIDIN-4-ONE AND THIENOPYRIDAZIN-7-ONE DERIVATIVES AS MCH RL ANTAGONISTS AstraZeneca AB (SE) 2009-11-25 EP disclosed
US-20080051405-A1 Therapeutic Agents ASTRAZENECA AB (SE) 2008-02-28 US disclosed
WO-2008020799-A1 THIENOPYRIMIDIN-4-ONE AND THIENOPYRIDAZIN-7-ONE DERIVATIVES AS MCH RL ANTAGONISTS ASTRAZENECA AB (SE) 2008-02-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080051405-A1 Therapeutic Agents GPR119, HTT, IAPP MGLL 509/4885GPR119 1/4885MDM2 4413/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.