SCHEMBL360334

SCHEMBL360334

Cc1c2cccc(C(N)=O)c2nn1C1CCCCN1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 15/20 0.47
PARP2 Q9UGN5 4/20 0.42
PARP3 Q9Y6F1 1/20 0.42
CD38 P28907 1/20 0.41
RPS6KB1 P23443 4/20 0.39
AURKA O14965 3/20 0.39
MAP4K4 O95819 1/20 0.39
CSF1R P07333 1/20 0.39
PIM1 P11309 1/20 0.39
CLK2 P49760 1/20 0.39
MAP4K2 Q12851 1/20 0.39
DYRK1A Q13627 1/20 0.39
MINK1 Q8N4C8 1/20 0.39
AURKB Q96GD4 1/20 0.39
MAP4K5 Q9Y4K4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL359495 0.97 PARP1 (0.46) PARP1PARP2PARP3CD38RPS6KB1
SCHEMBL12503403 0.90 PARP1 (0.36) PARP1PARP2PARP3RPS6KB1AURKA
SCHEMBL359578 0.86 PARP1 (0.47) PARP1PARP2PARP3CD38RPS6KB1
SCHEMBL12503322 0.86 PARP1 (0.39) PARP1PARP2PARP3RPS6KB1AURKA
SCHEMBL361151 0.84 PARP1 (0.45) PARP1PARP2PARP3RPS6KB1AURKA
SCHEMBL359562 0.84 PARP1 (0.32) PARP1CD38
SCHEMBL358329 0.83 PARP1 (0.46) PARP1PARP2PARP3RPS6KB1AURKA
SCHEMBL358843 0.81 PARP1 (0.44) PARP1PARP2PARP3RPS6KB1AURKA
SCHEMBL358368 0.81 RAD52 (0.45) PARP1
SCHEMBL358998 0.81 SCN4A (0.34) PARP1PARP2PARP3RPS6KB1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO claimed
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed