SCHEMBL3604381

SCHEMBL3604381

Brc1cc(Br)c(Br)s1.Fc1ccc(-c2cc(Br)c(-c3ccc(F)cc3)s2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SNCA P37840 1/20 0.44
PTGS2 P35354 3/20 0.40
PTGS1 P23219 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
KDM4E B2RXH2 2/20 0.40
MT-CO1 P00395 1/20 0.40
MT-CO2 P00403 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
IKBKB O14920 5/20 0.38
CHUK O15111 1/20 0.38
HSD17B1 P14061 1/20 0.34
HSD17B2 P37059 1/20 0.34
PTPN1 P18031 1/20 0.34
ESR1 P03372 2/20 0.33
ESR2 Q92731 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3613642 0.90 IKBKB (0.38) SNCAPTGS2PTGS1CYP1A2CYP3A4
SCHEMBL3597485 0.88 SNCA (0.53) SNCAPTGS2PTGS1CYP1A2CYP3A4
SCHEMBL3594365 0.83 IKBKB (0.42) SNCAPTGS2PTGS1CYP1A2CYP3A4
SCHEMBL23448488 0.71 SNCA (0.53) SNCACYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL14832796 0.71 SNCA (0.53) SNCAPTGS2CYP1A2KDM4EIKBKB
SCHEMBL16024135 0.70 SNCA (0.53) SNCAESR1ESR2
SCHEMBL915201 0.70 SNCA (0.52) SNCACYP1A2CYP3A4CYP2C9KDM4E
SCHEMBL27797494 0.69 IKBKB (0.40) SNCAPTGS2PTGS1CYP1A2CYP3A4
SCHEMBL917122 0.69
SCHEMBL3601307 0.68 PTPN1 (0.58) CYP1A2CYP3A4CYP2C9CYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8835476-B2 Synthesis of novel antimicrobials WU FAN (CA) 2014-09-16 US disclosed
US-20100076028-A1 Design and Synthesis of Novel Antimicrobials WU FAN 2010-03-25 US disclosed
WO-2006092059-A1 DESIGN AND SYNTHESIS OF NOVEL ANTIMICROBIALS WU FAN (CA) 2006-09-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100076028-A1 Design and Synthesis of Novel Antimicrobials MLX, LPXN, TPX2 SNCA 3933/4885PTGS2 2089/4885PTGS1 1164/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.