SCHEMBL3606671

SCHEMBL3606671

Cc1cc2ccc(CN)cc2s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.47
ROCK1 Q13464 2/20 0.38
ASIC3 Q9UHC3 2/20 0.36
LOXL2 Q9Y4K0 2/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA3 P07451 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8189102 0.82 SMN1; SMN2 (0.47) CYP2A6NPC1RAB9ASMN1; SMN2HDAC3
SCHEMBL3597089 0.81 HSD17B10 (0.50) CYP2A6CA12CA2CA3CA4
SCHEMBL24297526 0.78 ESR1 (0.38) NPC1RAB9ASMN1; SMN2HDAC3HDAC4
SCHEMBL19756719 0.78 CA2 (0.44) CA2HDAC3HDAC4HDAC1HDAC7
SCHEMBL8221541 0.78 GABRA1 (0.41) SMN1; SMN2HDAC3HDAC4HDAC1HDAC7
SCHEMBL422041 0.77 HDAC3 (0.52) CYP2A6NPC1RAB9AHDAC3HDAC4
SCHEMBL12278184 0.74 CA2 (0.52) CA1CA2CA4NPC1RAB9A
SCHEMBL1888634 0.72 PTPN2 (0.47) NPC1RAB9ASMN1; SMN2HDAC3HDAC4
SCHEMBL18949250 0.72 PTGS1 (0.41) NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL6232099 0.71 CYP2A6 (0.59) CYP2A6ROCK1ASIC3LOXL2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100298314-A1 NOVEL JNK INHIBITORS SCHERING CORPORATION 2010-11-25 US disclosed
EP-2134713-A2 NOVEL JNK INHIBITORS SCHERING CORPORATION (US) 2009-12-23 EP disclosed
WO-2008082490-A2 NOVEL JNK INHIBITORS SCHERING CORPORATION (US) 2008-07-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100298314-A1 NOVEL JNK INHIBITORS MAPK1, MAPKAPK2, MAP4K2 CYP2A6 1718/4885ROCK1 868/4885ASIC3 4694/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.